SCHEMBL6272298

SCHEMBL6272298

CCOC(=O)C1CCN(C(=O)COc2ccc3c(c2)OCO3)CC1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.63
MAPK1 P28482 2/20 0.63
TP53 P04637 1/20 0.63
MAPT P10636 1/20 0.63
FKBP1A P62942 1/20 0.63
KMT2A Q03164 3/20 0.62
POLB P06746 4/20 0.62
NPC1 O15118 2/20 0.62
RAB9A P51151 2/20 0.62
SMN1; SMN2 Q16637 2/20 0.57
HSD17B10 Q99714 1/20 0.57
ALDH1A1 P00352 4/20 0.57
MEN1 O00255 2/20 0.57
HPGD P15428 1/20 0.55
PKM P14618 1/20 0.55
LMNA P02545 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271302 0.83 POLB (0.66) KMT2APOLBNPC1RAB9AHSD17B10
SCHEMBL8145757 0.81 HPGD (0.77) TSHRKMT2APOLBNPC1RAB9A
SCHEMBL5533520 0.77 ALDH1A1 (0.66) MAPTFKBP1AKMT2ANPC1RAB9A
SCHEMBL8884329 0.76 KMT2A (0.66) TSHRMAPK1TP53MAPTKMT2A
SCHEMBL17541648 0.76 OGA (0.60) TSHRPOLBNPC1RAB9AALDH1A1
SCHEMBL8410149 0.72 ALDH1A1 (0.69) TSHRMAPK1TP53MAPTKMT2A
SCHEMBL6269813 0.72 ALDH1A1 (0.71) TSHRKMT2APOLBNPC1RAB9A
SCHEMBL2607028 0.71 POLB (0.65) TSHRMAPK1TP53MAPTKMT2A
SCHEMBL8389779 0.71 MAPT (0.62) TSHRMAPTFKBP1AKMT2APOLB
SCHEMBL6983366 0.71 ALDH1A1 (0.68) TSHRMAPK1TP53MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000620-B1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBITORS TAIHO PHARMACEUTICAL CO LTD (JP) 2005-12-07 EP disclosed
US-6166036-A Lp(a)-lowering agent and apolipoprotein (a) formation suppressing agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-26 US disclosed
EP-1000620-A1 Lp(a)-LOWERING AGENTS AND APOPROTEIN (a) PRODUCTION INHIBTORS TAIHO PHARMACEUTICAL COMPANY, LIMITED (JP) 2000-05-17 EP disclosed
EP-0393607-B1 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMA CO LTD (JP) 1996-02-21 EP disclosed
US-5145865-A Fatty acid, cholesterol synthesis inhibitors; enzyme inhibitors; antilipemic agents OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1992-09-08 US disclosed
EP-0393607-A2 Phenylcarboxylic acid derivatives having a hetero ring OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-10-24 EP disclosed