SCHEMBL6274175

SCHEMBL6274175

C=C(C)c1ccnc(/C=C/c2ccc(-c3nnn(COCC[Si](C)(C)C)n3)cc2)c1OCc1cccc(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.42
MMP13 P45452 2/20 0.36
RAB9A P51151 3/20 0.35
NPC1 O15118 2/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 2/20 0.34
USP2 O75604 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAOB P27338 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
RECQL P46063 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6274180 1.00 THRB (0.42) THRBMMP13RAB9ANPC1MAPT
SCHEMBL6272560 0.91 THRB (0.45) THRBMMP13RAB9ANPC1MAPT
SCHEMBL6278229 0.79 CD74 (0.33) THRBRAB9ANPC1MAPTALDH1A1
SCHEMBL6273142 0.76 SNCA (0.39) RAB9ANPC1MAPTALDH1A1KDM4E
SCHEMBL6273143 0.76 SNCA (0.39) RAB9ANPC1MAPTALDH1A1KDM4E
SCHEMBL6274709 0.67 MAPT (0.46) MAPTSMN1; SMN2MAOB
SCHEMBL6275956 0.65 NPC1 (0.46) RAB9ANPC1MAPTSMN1; SMN2HPGD
SCHEMBL6275960 0.65 NPC1 (0.46) RAB9ANPC1MAPTSMN1; SMN2HPGD
SCHEMBL6281046 0.62 MAOB (0.33) MAOB
SCHEMBL1058756 0.61 NPC1 (0.52) RAB9ANPC1MAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005116010-A1 EP4 RECEPTOR AGONIST, COMPOSITIONS AND METHODS THEREOF MERCK FROSST CANADA LTD. (CA) 2005-12-08 WO disclosed