SCHEMBL6281046

SCHEMBL6281046

COc1cccc(COc2c(C(C)C)ccnc2C=Cc2ccc(-c3nnn[nH]3)cc2)c1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.33
CHEK1 O14757 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCNA2 P20248 1/20 0.33
CCND1 P24385 1/20 0.33
CDK2 P24941 1/20 0.33
CCND3 P30281 1/20 0.33
NT5E P21589 1/20 0.33
MPO P05164 1/20 0.33
PIN1 Q13526 1/20 0.33
PLA2G2A P14555 1/20 0.32
AKR1C3 P42330 1/20 0.32
GLA P06280 2/20 0.32
IDO1 P14902 1/20 0.31
AGXT P21549 1/20 0.31
CDC25B P30305 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6276945 0.83 MAOB (0.38) MAOBMPO
SCHEMBL6275960 0.79 NPC1 (0.46) MAOBAKR1C3
SCHEMBL6275956 0.79 NPC1 (0.46) MAOBAKR1C3
SCHEMBL6281472 0.74 ABCB1 (0.33)
SCHEMBL6273406 0.71 MAPT (0.48) MAOBMPOIDO1AGXT
SCHEMBL6281237 0.69 ABCB1 (0.46) MAOB
SCHEMBL6279347 0.67 ABCB1 (0.40) MAOB
SCHEMBL8409057 0.67 HTR1A (0.37)
SCHEMBL6278229 0.66 CD74 (0.33) MAOBCDC25B
SCHEMBL6277363 0.66 CYP17A1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005116010-A1 EP4 RECEPTOR AGONIST, COMPOSITIONS AND METHODS THEREOF MERCK FROSST CANADA LTD. (CA) 2005-12-08 WO disclosed