SCHEMBL627431

SCHEMBL627431

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s1)CC2

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.48
HASPIN Q8TF76 7/20 0.42
KCNH2 Q12809 4/20 0.41
FLT3 P36888 4/20 0.41
KIT P10721 1/20 0.41
PIM1 P11309 1/20 0.41
CDK7 P50613 1/20 0.41
PIM3 Q86V86 1/20 0.41
PIM2 Q9P1W9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627019 0.94 PIK3CA (0.47) PIK3CAHASPINKCNH2FLT3KIT
SCHEMBL625421 0.92 PIK3CA (0.52) PIK3CAHASPINKCNH2FLT3KIT
SCHEMBL626122 0.91 PIK3CA (0.45) PIK3CAHASPINKCNH2FLT3KIT
SCHEMBL627432 0.87 RET (0.40) PIK3CA
SCHEMBL625407 0.85 PIK3CA (0.45) PIK3CAHASPIN
SCHEMBL627308 0.85 PIK3CA (0.49) PIK3CAKCNH2
SCHEMBL624438 0.83 PIK3CA (0.50) PIK3CAHASPINKCNH2FLT3KIT
SCHEMBL626245 0.83 PIK3CA (0.46) PIK3CAKCNH2
SCHEMBL627020 0.82 RET (0.40) PIK3CA
SCHEMBL625131 0.80 PIK3CA (0.49) PIK3CAHASPINKCNH2FLT3KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed