SCHEMBL627308

SCHEMBL627308

CC(C)(C)OC(=O)N1C[C@@H]2CN(c3nn4c(-c5cnc(N)c(C(F)(F)F)c5)cnc4s3)C[C@@H]2C1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.49
MAP3K12 Q12852 3/20 0.44
RIPK1 Q13546 2/20 0.40
USP30 Q70CQ3 1/20 0.39
KCNH2 Q12809 3/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625421 0.89 PIK3CA (0.52) PIK3CAMAP3K12RIPK1KCNH2
SCHEMBL627309 0.87 MAP3K12 (0.46) PIK3CAMAP3K12USP30
SCHEMBL626245 0.86 PIK3CA (0.46) PIK3CAMAP3K12RIPK1KCNH2
SCHEMBL627431 0.85 PIK3CA (0.48) PIK3CAKCNH2
SCHEMBL627019 0.84 PIK3CA (0.47) PIK3CAMAP3K12KCNH2HDAC1HDAC2
SCHEMBL626619 0.83 PIK3CA (0.55) PIK3CAMAP3K12KCNH2
SCHEMBL627310 0.82 PIK3CA (0.46) PIK3CAMAP3K12RIPK1
SCHEMBL626122 0.82 PIK3CA (0.45) PIK3CAKCNH2
SCHEMBL624990 0.80 PIK3CA (0.47) PIK3CARIPK1KCNH2
SCHEMBL625131 0.80 PIK3CA (0.49) PIK3CARIPK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed