SCHEMBL626207

SCHEMBL626207

CS(=O)(=O)N1CCC(Nc2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 6/20 0.46
CDK2 P24941 12/20 0.44
CCNE1 P24864 10/20 0.44
CCND1 P24385 9/20 0.42
CDK1 P06493 9/20 0.42
CDK4 P11802 8/20 0.42
CDK6 Q00534 7/20 0.42
CCNB1 P14635 7/20 0.42
CCND3 P30281 6/20 0.42
PIK3CA P42336 1/20 0.42
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625754 0.90 MAP3K12 (0.40) MAP3K12PIK3CA
SCHEMBL626704 0.87 CCNE1 (0.43) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL624428 0.87 MAP3K12 (0.47) MAP3K12PIK3CA
SCHEMBL624394 0.86 CCNE1 (0.41) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL625301 0.85 MAP3K12 (0.44) MAP3K12PIK3CA
SCHEMBL626206 0.84 PIK3CA (0.53) MAP3K12PIK3CA
SCHEMBL626165 0.84 IDO1 (0.47) CDK2CCNE1CCND1CDK1CDK4
SCHEMBL627397 0.84 PIK3CA (0.49) MAP3K12PIK3CA
SCHEMBL625456 0.84 MAP3K12 (0.41) MAP3K12CDK2CCNE1CCND1CDK1
SCHEMBL625236 0.84 MAP3K12 (0.45) MAP3K12PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed