SCHEMBL628002

SCHEMBL628002

CC1(O)CCC(Nc2nn3ccnc3s2)CC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 5/20 0.38
FYN P06241 6/20 0.36
KCNH2 Q12809 2/20 0.36
JAK1 P23458 4/20 0.34
JAK3 P52333 4/20 0.34
PIM2 Q9P1W9 2/20 0.34
CD38 P28907 2/20 0.34
TTK P33981 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
HPGDS O60760 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626162 0.79 CD38 (0.34) PIM1KCNH2CD38HPGDS
SCHEMBL627850 0.79 JAK1 (0.35) PIM1FYNKCNH2JAK1JAK3
SCHEMBL627849 0.77 FYN (0.46) PIM1FYNKCNH2JAK1JAK3
SCHEMBL626163 0.74 HSD11B1 (0.32) JAK1JAK3IRAK4
SCHEMBL625636 0.69 MAP3K12 (0.44)
SCHEMBL2250791 0.66 MKNK1 (0.53) PIM1FYNTTK
SCHEMBL12494024 0.63 IRAK4 (0.43) PIM1JAK1JAK3PIM2TTK
SCHEMBL2252121 0.61 MKNK1 (0.53) FYNTTK
SCHEMBL24765705 0.60 TTK (0.47) PIM1JAK1JAK3PIM2TTK
SCHEMBL25783428 0.60 TTK (0.47) PIM1JAK1JAK3PIM2TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed