SCHEMBL626162

SCHEMBL626162

CC1(O)CCC(NCc2nn3ccnc3s2)CC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CD38 P28907 2/20 0.34
PIM1 P11309 2/20 0.32
BMPR1B O00238 1/20 0.32
BMPR1A P36894 1/20 0.32
TGFBR1 P36897 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
GPX4 P36969 2/20 0.31
HPGDS O60760 2/20 0.31
ACKR3 P25106 1/20 0.31
NTRK1 P04629 1/20 0.31
KCNH2 Q12809 1/20 0.31
METTL3 Q86U44 1/20 0.30
VNN1 O95497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625008 0.79 PIM1 (0.35) PIM1BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL628002 0.79 PIM1 (0.38) CD38PIM1HPGDSKCNH2
SCHEMBL626163 0.71 HSD11B1 (0.32)
SCHEMBL625280 0.68 PIK3CA (0.49) PIM1BMPR1BBMPR1ATGFBR1ACVRL1
SCHEMBL2588468 0.63 OPRM1 (0.61)
SCHEMBL2250791 0.61 MKNK1 (0.53) PIM1
SCHEMBL24919667 0.60 KCNH2 (0.39) KCNH2
SCHEMBL18111942 0.60 KCNH2 (0.39) KCNH2
SCHEMBL20940105 0.60 KCNH2 (0.39) KCNH2
SCHEMBL627849 0.59 FYN (0.46) PIM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed