SCHEMBL6281472

SCHEMBL6281472

COc1cc(COc2c(C(C)C)ccnc2CCc2ccc(-c3nnn[nH]3)cc2)cc(OC)c1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.33
CYP19A1 P11511 1/20 0.32
CALM1 P0DP23 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6276945 0.92 MAOB (0.38) ABCB1
SCHEMBL6277363 0.88 CYP17A1 (0.31)
SCHEMBL6281809 0.87 ABCB1 (0.34) ABCB1CYP19A1
SCHEMBL6274623 0.87
SCHEMBL6277051 0.87 ABCB1 (0.34) ABCB1CYP19A1CALM1
SCHEMBL6274263 0.75
SCHEMBL6281046 0.74 MAOB (0.33)
SCHEMBL6274210 0.74 ABCB1 (0.38) ABCB1CYP19A1CALM1
SCHEMBL6281237 0.74 ABCB1 (0.46) ABCB1
SCHEMBL6278569 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005116010-A1 EP4 RECEPTOR AGONIST, COMPOSITIONS AND METHODS THEREOF MERCK FROSST CANADA LTD. (CA) 2005-12-08 WO claimed