SCHEMBL6276945

SCHEMBL6276945

COc1cccc(COc2c(C(C)C)ccnc2CCc2ccc(-c3nnn[nH]3)cc2)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.38
ABCB1 P08183 8/20 0.36
HTR1A P08908 3/20 0.36
DRD2 P14416 3/20 0.36
BRS3 P32247 1/20 0.34
MPO P05164 1/20 0.33
FLT1 P17948 1/20 0.33
KDR P35968 1/20 0.33
NR3C2 P08235 1/20 0.33
QPCTL Q9NXS2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6281472 0.92 ABCB1 (0.33) ABCB1
SCHEMBL6277363 0.84 CYP17A1 (0.31)
SCHEMBL6274623 0.83
SCHEMBL6281046 0.83 MAOB (0.33) MAOBMPO
SCHEMBL6281237 0.83 ABCB1 (0.46) MAOBABCB1HTR1ADRD2FLT1
SCHEMBL6281809 0.80 ABCB1 (0.34) ABCB1
SCHEMBL6277051 0.79 ABCB1 (0.34) ABCB1KDR
SCHEMBL6274294 0.79 MRGPRX4 (0.48) MAOB
SCHEMBL6274681 0.78 NR3C2 (0.43) MAOBNR3C2
SCHEMBL8409057 0.76 HTR1A (0.37) ABCB1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005116010-A1 EP4 RECEPTOR AGONIST, COMPOSITIONS AND METHODS THEREOF MERCK FROSST CANADA LTD. (CA) 2005-12-08 WO claimed