SCHEMBL628796

SCHEMBL628796

COc1ccc([C](CC(C)=O)c2ccc(OC)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.59
CA2 P00918 6/20 0.59
CES2 O00748 2/20 0.57
CES1 P23141 2/20 0.57
PLK1 P53350 1/20 0.55
PARP1 P09874 1/20 0.53
PARP10 Q53GL7 1/20 0.53
PARP2 Q9UGN5 1/20 0.53
PARP4 Q9UKK3 1/20 0.53
HDAC3 O15379 2/20 0.53
HDAC4 P56524 2/20 0.53
HDAC1 Q13547 2/20 0.53
HDAC7 Q8WUI4 2/20 0.53
HDAC2 Q92769 2/20 0.53
HDAC10 Q969S8 2/20 0.53
HDAC11 Q96DB2 2/20 0.53
HDAC8 Q9BY41 2/20 0.53
HDAC6 Q9UBN7 2/20 0.53
HDAC9 Q9UKV0 2/20 0.53
HDAC5 Q9UQL6 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1374066 0.84 ALDH1A1 (0.64) CA1CA2CES2CES1PLK1
P-Methoxy-Acetophenone SCHEMBL28038884 0.79 MAPT (0.55) CA1CA2CES2CES1PLK1
SCHEMBL11136993 0.79 ALDH1A1 (0.58) CA1CA2CES2CES1HDAC3
SCHEMBL153386 0.77 ALDH1A1 (0.76) CA1CA2CES2CES1PLK1
P-Methoxy-Acetophenone SCHEMBL41285 0.76 MAPT (0.70) CA1CA2CES2CES1PLK1
SCHEMBL5857541 0.76 NPC1 (0.65) CA1CA2PLK1NPC1RAB9A
SCHEMBL1987861 0.75 CA1 (0.61) CA1CA2CES2CES1PLK1
SCHEMBL6283202 0.74 MMP1 (0.67) CES2CES1HDAC3HDAC4HDAC1
P-Methoxy-Acetophenone SCHEMBL9835038 0.74 MAPT (0.67) CA1CA2CES2CES1PLK1
Methyl 4-Methoxybenzoate SCHEMBL231243 0.74 CA1 (1.00) CA1CA2CES2CES1PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1514542-B1 Medicinal composition comprising Tacrine or Donepezil for improving brain function. TOYAMA CHEMICAL CO LTD (JP) 2012-02-22 EP claimed