SCHEMBL628805

SCHEMBL628805

COC(=O)c1ccc(C(C)NCC2CCCCC2)cc1-c1ccccc1C

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.40
CNR1 P21554 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
MAPK14 Q16539 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL629208 0.99 BACE1 (0.40) BACE1CNR1ALDH1A1TSHR
SCHEMBL629649 0.83 FNTA (0.37)
SCHEMBL7870248 0.83 METAP2 (0.45) BACE1
SCHEMBL7870315 0.81 FNTA (0.54)
SCHEMBL7908810 0.80 FNTA (0.39) ALDH1A1
SCHEMBL628806 0.79 MEN1 (0.41)
SCHEMBL7874202 0.78 GCK (0.36)
Hydrochloric Acid SCHEMBL629209 0.78 MEN1 (0.41)
SCHEMBL7869097 0.78 NPC1 (0.56) BACE1
SCHEMBL628912 0.78 FNTA (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986384-B1 INHIBITORS OF PROTEIN ISOPRENYL TRANSFERASES UNIV PITTSBURGH (US) 2012-02-22 EP disclosed
US-6310095-B1 INHIBITING OR TREATING CANCER, TREATING INTIMAL HYPERPLASIA ASSOCIATED WITH RESTENOSIS AND ATHEROSCLEROSIS, INHIBITING POST-TRANSLATIONAL MODIFICATION OF ONCOGENIC RAS PROTEIN BY PROTEIN FARNESYLTRANSFERASE AND/OR GERANYLGERANYLTRANSFERASE UNIVERSITY OF PITTSBURGH 2001-10-30 US disclosed