SCHEMBL629270

SCHEMBL629270

COC(=O)c1ccc2c(c1)[nH]c(=O)c1ccncc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 1.00
CSNK2A1 P68400 4/20 1.00
DYRK1A Q13627 1/20 0.57
KIF11 P52732 2/20 0.56
ROCK2 O75116 2/20 0.54
ROCK1 Q13464 1/20 0.54
GSK3B P49841 1/20 0.51
CSNK2A2 P19784 1/20 0.50
CSNK2B P67870 1/20 0.50
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
GLA P06280 1/20 0.48
GAA P10253 1/20 0.48
PKM P14618 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
HSD17B10 Q99714 1/20 0.48
RAB9A P51151 1/20 0.48
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30704691 1.00 PARP1 (1.00) PARP1CSNK2A1DYRK1AKIF11ROCK2
SCHEMBL2691509 0.95 PARP1 (0.90) PARP1CSNK2A1DYRK1AKIF11ROCK2
SCHEMBL10134619 0.90 PARP1 (0.81) PARP1CSNK2A1DYRK1AKIF11ROCK2
SCHEMBL16377295 0.87 PARP1 (0.76) PARP1CSNK2A1DYRK1AKIF11ROCK2
SCHEMBL30172793 0.85 PARP1 (0.74) PARP1CSNK2A1DYRK1AKIF11ROCK2
SCHEMBL4972014 0.84 PARP1 (1.00) PARP1CSNK2A1DYRK1AROCK2ROCK1
SCHEMBL10135321 0.83 PARP1 (0.78) PARP1CSNK2A1ROCK2ROCK1GSK3B
SCHEMBL10134618 0.82 PARP1 (0.70) PARP1CSNK2A1DYRK1AROCK2ROCK1
SCHEMBL25293367 0.82 PARP1 (1.00) PARP1CSNK2A1DYRK1AKIF11KMT2A
SCHEMBL628532 0.80 PARP1 (0.67) PARP1CSNK2A1DYRK1AKIF11GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12383624-B2 Cargo delivery system and composition comprising the same SEOUL NATIONAL UNIVERSITY R&DB FOUNDATION (KR) 2025-08-12 US disclosed
CN-117263934-A Preparation method of 5H-benzo [ c ] [1,6] naphthyridine-6-ketone derivative 上海凌凯医药科技有限公司 2023-12-22 CN disclosed
WO-2023126951-A1 INHIBITORS OF AUTOPHAGY-RELATED PROTEIN-PROTEIN INTERACTIONS YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2023-07-06 WO disclosed
WO-2023126951-A1 INHIBITORS OF AUTOPHAGY-RELATED PROTEIN-PROTEIN INTERACTIONS YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2023-07-06 WO disclosed
US-20230190938-A1 NOVEL CARGO DELIVERY SYSTEM AND COMPOSITION COMPRISING THE SAME SEOUL NATIONAL UNIVERSITY R&DB FOUNDATION (KR) 2023-06-22 US disclosed
US-20230190938-A1 NOVEL CARGO DELIVERY SYSTEM AND COMPOSITION COMPRISING THE SAME SEOUL NATIONAL UNIVERSITY R&DB FOUNDATION (KR) 2023-06-22 US disclosed
US-11071727-B2 Therapeutic targeting of proteolytic cleavage of the mixed lineage leukemia gene product (MLL1) by taspase1 using kinase inhibitors NORTHWESTERN UNIVERSITY (US) 2021-07-27 US disclosed
US-20190231759-A1 THERAPEUTIC TARGETING OF PROTEOLYTIC CLEAVAGE OF THE MIXED LINEAGE LEUKEMIA GENE PRODUCT (MLL1) BY TASPASE1 USING KINASE INHIBITORS NORTHWESTERN UNIVERSITY (US) 2019-08-01 US disclosed
US-9176064-B2 Bisubstrate fluorescent probes for protein kinase CK2 UNIVERSITY OF TARTU (EE) 2015-11-03 US disclosed
US-9176064-B2 Bisubstrate fluorescent probes for protein kinase CK2 UNIVERSITY OF TARTU (EE) 2015-11-03 US disclosed
WO-2009097014-A2 THERAPEUTIC KINASE MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2009-08-06 WO disclosed
EP-2061765-A2 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS Cylene Pharmaceuticals, Inc. (US) 2009-05-27 EP disclosed
US-20090105233-A1 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS SENHWA BIOSCIENCES, INC. (TW) 2009-04-23 US disclosed
US-20090105233-A1 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS SENHWA BIOSCIENCES, INC. (TW) 2009-04-23 US disclosed
US-20090105233-A1 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS SENHWA BIOSCIENCES, INC. (TW) 2009-04-23 US disclosed
US-20090093465-A1 THERAPEUTIC KINASE MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2009-04-09 US disclosed
US-20090093465-A1 THERAPEUTIC KINASE MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2009-04-09 US disclosed
US-20090093465-A1 THERAPEUTIC KINASE MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2009-04-09 US disclosed
WO-2008028168-A2 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2008-03-06 WO disclosed
WO-2008028168-A2 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2008-03-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190231759-A1 THERAPEUTIC TARGETING OF PROTEOLYTIC CLEAVAGE OF THE MIXED LINEAGE LEUKEMIA GENE PRODUCT (MLL1) BY TASPASE1 USING KINASE INHIBITORS MLLT1, TASP1, MLLT3 PARP1 317/4885CSNK2A1 38/4885DYRK1A 1713/4885
US-20230190938-A1 NOVEL CARGO DELIVERY SYSTEM AND COMPOSITION COMPRISING THE SAME ATG7, SQSTM1, BECN1 PARP1 2432/4885CSNK2A1 956/4885DYRK1A 2472/4885
US-12383624-B2 Cargo delivery system and composition comprising the same ATG7, SQSTM1, BECN1 PARP1 2026/4885CSNK2A1 1104/4885DYRK1A 2481/4885
US-20090093465-A1 THERAPEUTIC KINASE MODULATORS PACSIN2, CKS1B, CSNK1A1 PARP1 1797/4885CSNK2A1 6/4885DYRK1A 427/4885
US-20090105233-A1 SERINE-THREONINE PROTEIN KINASE AND PARP MODULATORS PACSIN2, TNKS, PARP1 PARP1 3/4885CSNK2A1 24/4885DYRK1A 502/4885
US-11071727-B2 Therapeutic targeting of proteolytic cleavage of the mixed lineage leukemia gene product (MLL1) by taspase1 using kinase inhibitors MLLT1, TASP1, MLLT3 PARP1 317/4885CSNK2A1 38/4885DYRK1A 1713/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.