SCHEMBL6294474

SCHEMBL6294474

O=C(Cl)/C=C/c1cc2ccccc2o1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.62
MAPK1 P28482 3/20 0.62
MAPT P10636 2/20 0.62
NPC1 O15118 2/20 0.62
CYP2A6 P11509 1/20 0.56
PLIN1 O60240 1/20 0.52
LMNA P02545 1/20 0.52
GAA P10253 1/20 0.52
PLIN5 Q00G26 1/20 0.52
ABHD5 Q8WTS1 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
FLT3 P36888 1/20 0.47
APP P05067 1/20 0.47
MAOB P27338 4/20 0.44
TSHR P16473 2/20 0.42
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6294475 1.00 RAB9A (0.62) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL1226009 0.85 MAPT (0.64) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL1226012 0.85 MAPT (0.64) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL29871432 0.85 MAPT (0.64) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL9799652 0.83 MAPT (0.62) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL3209460 0.83 RAB9A (0.62) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL9799655 0.83 MAPT (0.62) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL3209446 0.83 RAB9A (0.62) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL30963012 0.83 MAPT (0.62) RAB9AMAPK1MAPTNPC1CYP2A6
SCHEMBL10554653 0.81 RAB9A (0.59) RAB9AMAPK1MAPTNPC1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023178040-A2 INHIBITORS OF EWS-FLI1 UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2023-09-21 WO disclosed
US-6936600-B2 Sorbitol dehrydrogenase inhibitors PFIZER INC (US) 2005-08-30 US disclosed
US-6869943-B2 Sorbitol dehydrogenase inhibitors PFIZER INC (US) 2005-03-22 US disclosed
US-20050020578-A1 Sorbitol dehydrogenase inhibitors PFIZER INC. 2005-01-27 US disclosed
US-20040077671-A1 Sorbitol dehydrogenase inhibitors CHU-MOYER MARGARET Y (US) 2004-04-22 US disclosed
US-6660740-B1 Sorbitol dehydrogenase inhibitors PFIZER INC 2003-12-09 US disclosed
US-6602875-B2 Sorbitol dehydrogenase inhibitors PFIZER INC 2003-08-05 US disclosed
US-20030065179-A1 Sorbitol dehydrogenase inhibitors CHU-MOYER MARGARET Y (US) 2003-04-03 US disclosed
US-6414149-B1 TREATING DIABETES, TREATING OR PREVENTING DIABETIC COMPLICATIONS PFIZER INC. 2002-07-02 US disclosed
EP-1185275-A1 AMINOPYRIMIDINES AS SORBITOL DEHYDROGENASE INHIBITORS Pfizer Products Inc. (US) 2002-03-13 EP disclosed
WO-2000059510-A1 AMINOPYRIMIDINES AS SORBITOL DEHYDROGENASE INHIBITORS PFIZER PRODUCTS INC. (US) 2000-10-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020578-A1 Sorbitol dehydrogenase inhibitors SLC5A1, SORD, SLC5A2 RAB9A 2713/4885MAPK1 792/4885MAPT 2491/4885
US-20040077671-A1 Sorbitol dehydrogenase inhibitors SLC5A1, SORD, SLC5A2 RAB9A 2389/4885MAPK1 799/4885MAPT 2399/4885
US-20030065179-A1 Sorbitol dehydrogenase inhibitors SLC5A1, SORD, SLC5A2 RAB9A 2389/4885MAPK1 799/4885MAPT 2399/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.