SCHEMBL6295705

SCHEMBL6295705

CCOC(=O)c1c(-c2ccccc2)[nH]c2ccc(OC)cc2c1=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.63
ALDH1A1 P00352 5/20 0.63
HPGD P15428 5/20 0.63
HSD17B10 Q99714 3/20 0.63
MAPT P10636 2/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
LMNA P02545 2/20 0.63
GAA P10253 1/20 0.63
MAPK10 P53779 1/20 0.63
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
TUBB4A P04350 1/20 0.55
TUBB P07437 1/20 0.55
TUBA3C P0DPH7 1/20 0.55
TUBA1B P68363 1/20 0.55
TUBA4A P68366 1/20 0.55
TUBB4B P68371 1/20 0.55
TUBB3 Q13509 1/20 0.55
TUBB2A Q13885 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300606 0.92 KDM4E (0.56) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6295726 0.89 ALDH1A1 (0.55) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6296000 0.88 KDM4E (0.54) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6294956 0.88 ALOX5 (0.66) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6295920 0.86 ALOX5 (0.57) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6294584 0.86 ALOX5 (0.57) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6300691 0.86 TUBB4A (0.62) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6300719 0.85 ALDH1A1 (0.67) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6295725 0.85 CSF1R (0.71) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL6294686 0.85 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897316-B2 Substituted 2-phenyl-4-quinolone-3-carboxylic acid compounds and their use as antitumor agents CHINA MEDICAL UNIVERSITY (TW) 2005-05-24 US disclosed
US-20050032832-A1 Substituted 2-phenyl-4-quinolone-3-carboxylic acid compounds and their use as antitumor agents CHINA MEDICAL UNIVERSITY (TW) 2005-02-10 US disclosed
EP-0785191-B1 FUSED INDAN DERIVATIVES AND SALTS THEREOF TAIHO PHARMACEUTICAL CO LTD (JP) 2002-10-23 EP disclosed
US-5763453-A ANTITUMOR AGENTS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-06-09 US disclosed
EP-0785191-A1 FUSED INDAN DERIVATIVES AND SALTS THEREOF TAIHO PHARMACEUTICAL CO., LTD. (JP) 1997-07-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050032832-A1 Substituted 2-phenyl-4-quinolone-3-carboxylic acid compounds and their use as antitumor agents TP53, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CHUK KDM4E 1042/4885ALDH1A1 465/4885HPGD 1434/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.