SCHEMBL630070

SCHEMBL630070

CC(C)(C)C(=O)N[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCCCN1S(=O)(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 7/20 0.56
ITGB1 P05556 3/20 0.51
ITGA5 P08648 2/20 0.51
PKM P14618 2/20 0.51
ALDH1A1 P00352 3/20 0.50
LMNA P02545 3/20 0.50
MAPK1 P28482 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
POLB P06746 1/20 0.49
CCR4 P51679 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
USP2 O75604 1/20 0.48
MAPT P10636 1/20 0.48
HSD17B10 Q99714 1/20 0.48
AKR1C3 P42330 1/20 0.47
GLA P06280 1/20 0.47
HTT P42858 1/20 0.47
ITGA4 P13612 1/20 0.46
ITGA2 P17301 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1384306 1.00 FKBP1A (0.56) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL630023 0.85 AKR1C3 (0.44) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL630983 0.85 CCR4 (0.53) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL1381491 0.85 CCR4 (0.53) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL630215 0.83 FKBP1A (0.53) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL1383786 0.83 FKBP1A (0.53) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL630190 0.82 FKBP1A (0.53) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL1380441 0.82 FKBP1A (0.53) FKBP1AITGB1ITGA5PKMALDH1A1
SCHEMBL1381163 0.81 MMP1 (0.55) FKBP1AITGB1ITGA5LMNATDP1
SCHEMBL629854 0.81 MMP1 (0.55) FKBP1AITGB1ITGA5LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778637-B1 FKBP-binding composition and pharmaceutical use thereof AVENTIS PHARMA INC (US) 2012-02-22 EP claimed
JP-4812758-B2 2011-11-09 JP claimed
EP-1778637-B1 FKBP-binding composition and pharmaceutical use thereof AVENTIS PHARMA INC (US) 2012-02-22 EP disclosed