SCHEMBL630084

SCHEMBL630084

N#Cc1ccc(N)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.52
IMPDH1 P20839 2/20 0.52
AR P10275 5/20 0.47
IDO1 P14902 2/20 0.46
EP300 Q09472 2/20 0.46
KAT8 Q9H7Z6 2/20 0.46
HDAC3 O15379 1/20 0.46
KAT2B Q92831 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
ALDH1A1 P00352 3/20 0.46
CYP3A4 P08684 3/20 0.46
HPGD P15428 2/20 0.46
TSHR P16473 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30175215 1.00 IMPDH2 (0.52) IMPDH2IMPDH1ARIDO1EP300
SCHEMBL19072727 0.94 AR (0.47) IMPDH2IMPDH1ARIDO1EP300
SCHEMBL30881802 0.86 ALDH1A1 (0.59) IMPDH2IMPDH1ARIDO1ALDH1A1
SCHEMBL4085978 0.86 ALDH1A1 (0.59) IMPDH2IMPDH1ARIDO1ALDH1A1
SCHEMBL31588265 0.86 ALDH1A1 (0.59) IMPDH2IMPDH1ARIDO1ALDH1A1
SCHEMBL29489135 0.85 IMPDH2 (0.64) IMPDH2IMPDH1ARALDH1A1TSHR
SCHEMBL151936 0.85 IMPDH2 (0.64) IMPDH2IMPDH1ARALDH1A1TSHR
SCHEMBL6650616 0.83 SLC22A12 (0.43) IMPDH2IMPDH1ARIDO1EP300
SCHEMBL11193357 0.83 IMPDH2 (0.61) IMPDH2IMPDH1ARALDH1A1TSHR
SCHEMBL11228244 0.80 IMPDH2 (0.59) IMPDH2IMPDH1ARALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 295 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734671-A Benzimidazoles derivative, preparation method and application 北京医药集团有限责任公司 2019-05-10 CN claimed
CN-107400090-A A kind of synthetic method of benzimidizole derivatives 华润赛科药业有限责任公司 2017-11-28 CN claimed
US-9194807-B2 Multi-layered devices for analyte detection KIMBERLY-CLARK WORLDWIDE, INC. (US) 2015-11-24 US claimed
US-20150260658-A1 Multi-Layered Devices for Analyte Detection KIMBERLY CLARK CO (US) 2015-09-17 US claimed
EP-2220250-B1 MULTI-LAYERED DEVICES FOR ANALYTE DETECTION KIMBERLY CLARK CO (US) 2014-09-03 EP claimed
CN-101896621-B Multi-layered device for analyte detection KIMBERLY CLARK CO 2014-05-14 CN claimed
US-8003399-B2 Nitrite detection technique KIMBERLY-CLARK WORLDWIDE, INC. (US) 2011-08-23 US claimed
EP-1920251-B1 NITRITE DETECTION TECHNIQUE KIMBERLY CLARK CO (US) 2010-12-29 EP claimed
CN-101896621-A Multi-layered device for analyte detection KIMBERLY CLARK CO 2010-11-24 CN claimed
US-20100290948-A1 ABSORBENT ARTICLES CAPABLE OF INDICATING THE PRESENCE OF URINARY TRACT INFECTIONS KIMBERLY-CLARK WORLDWIDE, INC. 2010-11-18 US claimed
WO-2009077886-A1 MULTI-LAYERED DEVICES FOR ANALYTE DETECTION KIMBERLY-CLARK WORLDWIDE, INC. (US) 2009-06-25 WO claimed
US-20090155122-A1 Multi-Layered Devices for Analyte Detection KIMBERLY-CLARK WORLDWIDE, INC. (US) 2009-06-18 US claimed
EP-1920251-A1 NITRITE DETECTION TECHNIQUE Kimberly-Clark Worldwide, Inc. (US) 2008-05-14 EP claimed
WO-2007027198-A1 NITRITE DETECTION TECHNIQUE KIMBERLY-CLARK WORLDWIDE, INC. (US) 2007-03-08 WO claimed
US-20070048182-A1 Nitrite detection technique KIMBERLY-CLARK WORLDWIDE, INC. 2007-03-01 US claimed
EP-0515379-A4 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INC (US) 1994-09-14 EP claimed
EP-0515379-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1992-12-02 EP claimed
US-5094740-A TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED, INC. (US) 1992-03-10 US claimed
WO-1991012276-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1991-08-22 WO claimed
WO-1991012275-A1 TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED INCORPORATED (US) 1991-08-22 WO claimed