SCHEMBL6304263

SCHEMBL6304263

CCCc1nc2cc(Cl)c(Cl)cc2nc1[S+]([O-])c1nnnn1C

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 1/20 0.40
GAA P10253 1/20 0.31
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6305850 0.70 GLP1R (0.41) GLP1R
SCHEMBL6307488 0.69 GLP1R (0.59) GLP1RGAA
SCHEMBL6304446 0.63 ALDH1A1 (0.46) GAA
SCHEMBL14486902 0.63 ALDH1A1 (0.41)
SCHEMBL16526249 0.58 ALDH1A1 (0.36)
SCHEMBL6303925 0.58 GLP1R (1.00) GLP1R
SCHEMBL6312923 0.56 GLP1R (0.71) GLP1R
SCHEMBL11116507 0.56 ALDH1A1 (0.39)
SCHEMBL10975195 0.56 ALDH1A1 (0.39)
SCHEMBL11870814 0.55 CUL4A (0.50) GAAHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6927214-B1 Non-peptide GLP-1 agonists NOVO NORDISK A/S (DK) 2005-08-09 US disclosed
EP-1147094-A1 NON-PEPTIDE GLP-1 AGONISTS NOVO NORDISK A/S (DK) 2001-10-24 EP disclosed
WO-2000042026-A1 NON-PEPTIDE GLP-1 AGONISTS NOVO NORDISK A/S (DK) 2000-07-20 WO disclosed