SCHEMBL6305993

SCHEMBL6305993

COc1ccc(-c2ccc(-c3nc4ccc(Cl)cc4c(=O)n3Cc3cccc(CN)c3)cc2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
F11 P03951 2/20 0.48
POLB P06746 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
ALDH1A1 P00352 6/20 0.45
USP2 O75604 3/20 0.45
TP53 P04637 3/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 3/20 0.45
LMNA P02545 2/20 0.45
HSD17B10 Q99714 2/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2B Q13224 1/20 0.45
MAPK1 P28482 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
BRD4 O60885 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6308119 0.94 F11 (0.52) TSHRF11ALDH1A1TP53LMNA
SCHEMBL6309689 0.93 F11 (0.48) TSHRF11POLBRXFP1ALDH1A1
SCHEMBL6313772 0.92 F11 (0.49) TSHRF11ALDH1A1LMNAGRIN1
SCHEMBL6313234 0.91 F11 (0.52) TSHRF11POLBRXFP1ALDH1A1
SCHEMBL6309491 0.90 F11 (0.60) TSHRF11POLBRXFP1ALDH1A1
SCHEMBL7551450 0.89 USP2 (0.46) TSHRF11POLBRXFP1ALDH1A1
SCHEMBL7549261 0.88 TSHR (0.43) TSHRPOLBRXFP1ALDH1A1USP2
SCHEMBL6306228 0.87 POLB (0.50) TSHRF11POLBRXFP1ALDH1A1
SCHEMBL6308212 0.87 F11 (0.52) TSHRF11POLBRXFP1ALDH1A1
SCHEMBL7551638 0.86 F11 (0.47) TSHRF11ALDH1A1TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed