SCHEMBL6306594

SCHEMBL6306594

COCS[PH](=O)Cc1ccc2cccc(C(=O)OC(C)(C)C)c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.37
NQO2 P16083 1/20 0.33
MTNR1A P48039 1/20 0.33
CACNA1B Q00975 1/20 0.33
APBA1 Q02410 1/20 0.33
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
CDC25B P30305 1/20 0.32
SLC7A5 Q01650 1/20 0.31
NR1H2 P55055 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 2/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
CRHBP P24387 1/20 0.30
CRHR2 Q13324 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6304064 0.77 NQO2 (0.39) CNR2NQO2MTNR1ACACNA1BAPBA1
SCHEMBL6306590 0.74 MTNR1A (0.37) CNR2NQO2MTNR1ACACNA1BAPBA1
SCHEMBL6303858 0.73 CNR2 (0.38) CNR2NQO2MTNR1ACACNA1BAPBA1
SCHEMBL6306592 0.73 MTNR1A (0.36) CNR2NQO2MTNR1ACACNA1BAPBA1
SCHEMBL6306600 0.72 NQO2 (0.33) NQO2MTNR1AADRB2ADRB1ADRB3
SCHEMBL974720 0.69 NR4A1 (0.53) ADRB2ADRB1ADRB3CDC25BKDM4E
SCHEMBL1204440 0.68 KDM4E (0.56) MTNR1AADRB2ADRB1ADRB3CDC25B
SCHEMBL6235824 0.67 CYP4F2 (0.38) CACNA1BAPBA1ADRB2ADRB1ADRB3
SCHEMBL31395544 0.67 KDM4E (0.54) MTNR1AADRB2ADRB1ADRB3CDC25B
SCHEMBL14627192 0.66 AR (0.41) ADRB2ADRB1ADRB3CDC25BSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6943267-B1 compounds structurally resemble the substrates of the enzymes, but have nonhydrolyzable mono protonated thiophosphonate salts; chromatography or distillations not required UTAH STATE UNIVERSITY (US) 2005-09-13 US disclosed
US-20050049431-A1 Thiophosphonate inhibitors of phosphatase enzymes and metallophosphatases UTAH STATE UNIVERSITY 2005-03-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050049431-A1 Thiophosphonate inhibitors of phosphatase enzymes and metallophosphatases PPME1, MTMR1, PTPRE CNR2 4521/4885NQO2 945/4885MTNR1A 2182/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.