SCHEMBL6309074

SCHEMBL6309074

CCN(CC)CCn1c(-c2ccccc2)nc2c(Cl)cc(Cl)cc2c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 12/20 0.48
KDM4E B2RXH2 9/20 0.48
HSD17B10 Q99714 9/20 0.48
HPGD P15428 8/20 0.48
TSHR P16473 8/20 0.48
CYP3A4 P08684 7/20 0.48
MAPT P10636 1/20 0.47
CASP1 P29466 1/20 0.46
EGFR P00533 1/20 0.46
FABP4 P15090 1/20 0.45
FABP5 Q01469 1/20 0.45
ALOX15 P16050 1/20 0.45
TOP2A P11388 1/20 0.44
BCL2 P10415 1/20 0.43
MCL1 Q07820 1/20 0.43
RAD52 P43351 2/20 0.43
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6309405 0.91 MEN1 (0.60) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL6306872 0.89 MEN1 (0.50) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL6310437 0.87 ALDH1A1 (0.52) ALDH1A1KDM4EHSD17B10HPGDTSHR
SCHEMBL6306022 0.84 EGFR (0.58) MEN1KMT2AALDH1A1KDM4ETSHR
SCHEMBL6309585 0.83 MEN1 (0.48) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL6308896 0.82 MEN1 (0.50) MEN1KMT2AALDH1A1KDM4EMAPT
SCHEMBL7549017 0.81 MEN1 (0.49) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL6307702 0.80 MEN1 (0.62) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL6308959 0.79 ABCC1 (0.47) MEN1KMT2AALDH1A1KDM4EHSD17B10
SCHEMBL7550755 0.79 CASR (0.64) MEN1KMT2AALDH1A1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed