SCHEMBL6310050

SCHEMBL6310050

CC1Oc2ccc(C(N)(CCCNC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)cc2N=C1N

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.34
CA2 P00918 8/20 0.34
CA12 O43570 4/20 0.34
CA9 Q16790 4/20 0.34
MIF P14174 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
BRD4 O60885 2/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2A1 P68400 1/20 0.31
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP1A1 P04798 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5466884 0.87 CA14 (0.32) MEN1KMT2A
SCHEMBL6281732 0.86
SCHEMBL5473214 0.84 DRD2 (0.30) DRD2
SCHEMBL6310057 0.81
SCHEMBL6303014 0.76
SCHEMBL6310051 0.76 CA14 (0.36) CA1CA2CA12CA9MIF
SCHEMBL6310004 0.73
SCHEMBL7708015 0.73 AAK1 (0.32) CCNCCDK8
SCHEMBL7710854 0.73
SCHEMBL7708340 0.72 ALDH1A1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6841550-B1 Benzoxazine and benzothiazine derivatives and their use in medicines SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-11 US disclosed
EP-1114037-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AG (DE) 2004-05-12 EP disclosed