SCHEMBL7708015

SCHEMBL7708015

CC1Oc2ccc(C(C)(NC(=O)OC(C)(C)C)c3ccncc3)cc2N=C1N

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.32
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
HASPIN Q8TF76 1/20 0.31
CDK19 Q9BWU1 1/20 0.31
CYP17A1 P05093 2/20 0.31
LATS1 O95835 1/20 0.30
KDM4D Q6B0I6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711071 0.89 NAMPT (0.36) CCNCCDK8HASPINCDK19CYP17A1
SCHEMBL7710854 0.86
SCHEMBL7711556 0.86 NPC1 (0.33)
SCHEMBL7708340 0.85 ALDH1A1 (0.32)
SCHEMBL7705092 0.82 NPSR1 (0.36)
SCHEMBL7711103 0.80 SMYD3 (0.39) LATS1
SCHEMBL7094003 0.80 ADORA2B (0.32) AAK1CYP17A1LATS1KDM4D
SCHEMBL7708011 0.75 LATS1 (0.34) AAK1CYP17A1LATS1
SCHEMBL7704894 0.73 CTSK (0.31)
SCHEMBL6310050 0.73 CA1 (0.34) CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed