SCHEMBL6312002

SCHEMBL6312002

OCc1cccc(CC2COCC(SC3COCC(c4cccc(CO)c4)O3)O2)c1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.34
CHRM4 P08173 4/20 0.34
CHRM5 P08912 4/20 0.34
CHRM1 P11229 4/20 0.34
CHRM3 P20309 3/20 0.34
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
HTR1A P08908 2/20 0.30
ADRA1D P25100 2/20 0.30
ADRA1A P35348 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6197809 0.73 CHRNB4 (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL6794902 0.68 HTR1A (0.36) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL6405563 0.68 CHRNB4 (0.34) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL22325696 0.68 ENPP2 (0.40) CHRNB4CHRNA3
SCHEMBL18890109 0.68 DRD2 (0.48) CHRNB4CHRNA3DRD2DRD3
SCHEMBL3767767 0.67 CHRNB4 (0.40) CHRNB4CHRNA3DRD2DRD3HTR1A
SCHEMBL19101551 0.65 TSHR (0.47) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL758717 0.62 ENPP2 (0.44) CHRNB4CHRNA3
SCHEMBL15698942 0.60 CHRM2 (0.62) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL23647871 0.60 DRD2 (0.47) CHRNB4CHRNA3DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1680338-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-10-12 CN disclosed
US-6867203-B2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2005-03-15 US disclosed
CN-1192018-C Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2005-03-09 CN disclosed
EP-1481968-A2 Cell adhesion-inhibiting anti-inflammatory and immune-suppressive compounds Abbott Laboratories (US) 2004-12-01 EP disclosed
US-20040116518-A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES 2004-06-17 US disclosed
CN-1350520-A Anti-inflammatory and immunosuppressive cell adhesion inhibiting compounds ABBOTT LAB (US) 2002-05-22 CN disclosed
EP-1140814-A2 CELL ADHESION-INHIBITING ANTIINFLAMMATORY AND IMMUNE-SUPPRESSIVE COMPOUNDS ABBOTT LABORATORIES (US) 2001-10-10 EP disclosed
WO-2000039081-A2 CELL ADHESION-INHIBITING ANTIINFLAMMATORY AND IMMUNE-SUPPRESSIVE COMPOUNDS ABBOTT LABORATORIES (US) 2000-07-06 WO disclosed