SCHEMBL6313330

SCHEMBL6313330

[CH2]c1ccc2cc(-c3ccccc3)ccc2c1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.49
GRIN2A Q12879 1/20 0.49
GRIN2B Q13224 1/20 0.49
GRIN2C Q14957 1/20 0.49
HSD17B1 P14061 5/20 0.49
HSD17B2 P37059 5/20 0.49
ESR1 P03372 6/20 0.49
ESR2 Q92731 6/20 0.49
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
GPR84 Q9NQS5 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2B6 P20813 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6318709 0.80 ESR1 (0.58) GRIN2DGRIN2AGRIN2BGRIN2CHSD17B1
SCHEMBL1527510 0.80 GRIN2D (0.54) GRIN2DGRIN2AGRIN2BGRIN2CHSD17B1
SCHEMBL6313341 0.79 GRIN2D (0.49) GRIN2DGRIN2AGRIN2BGRIN2CHSD17B1
SCHEMBL19501075 0.79 ESR2 (0.77) GRIN2DGRIN2AGRIN2BGRIN2CHSD17B1
SCHEMBL1987912 0.78 ESR1 (0.58) HSD17B1HSD17B2ESR1ESR2GPR84
SCHEMBL30703158 0.78 ESR1 (0.58) HSD17B1HSD17B2ESR1ESR2GPR84
SCHEMBL2724557 0.78 ESR1 (0.58) HSD17B1HSD17B2ESR1ESR2GPR84
SCHEMBL25825360 0.78 GRIN2D (0.55) GRIN2DGRIN2AGRIN2BGRIN2CHSD17B1
SCHEMBL3005121 0.76 ESR1 (0.56) HSD17B1HSD17B2ESR1ESR2GPR84
SCHEMBL21124585 0.76 ALDH1A1 (0.54) GRIN2DGRIN2AGRIN2BGRIN2CHSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217942-C Pyrrolidine derivatives having phospholipase A inhibitory activity SHIONOGI & CO (JP) 2005-09-07 CN disclosed
CN-1217699-C Preventives or remedies for arrhythmia SHIONOGI & CO (JP) 2005-09-07 CN disclosed
US-6924301-B1 Composition for treating or preventing arrhythmia SHIONOGI & CO., LTD. (JP) 2005-08-02 US disclosed
EP-0976748-B1 PYRROLIDINE DERIVATIVES HAVING PHOSPHOLIPASE A2 INHIBITORY ACTIVITY SHIONOGI & CO (JP) 2003-12-03 EP disclosed
CN-1411379-A Preventives or remedies for arrhythmia SHIONOGI & CO (JP) 2003-04-16 CN disclosed
EP-1240906-A1 PREVENTIVES OR REMEDIES FOR ARRHYTHMIA SHIONOGI & CO., LTD. (JP) 2002-09-18 EP disclosed
US-6147100-A ANTIINFLAMMATORY AGENTS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
CN-1251587-A Pyrrolidine derivatives having phospholipase A inhibitory activity SHIONOGI & CO (JP) 2000-04-26 CN disclosed
EP-0976748-A1 PYRROLIDINE DERIVATIVES HAVING PHOSPHOLIPASE A2 INHIBITORY ACTIVITY SHIONOGI & CO., LTD. (JP) 2000-02-02 EP disclosed