SCHEMBL6313852

SCHEMBL6313852

COc1ccc(-c2nc3cc(Cl)ccc3c(=O)n2CCCN)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.64
POLB P06746 3/20 0.54
RXFP1 Q9HBX9 2/20 0.54
ALDH1A1 P00352 5/20 0.52
MAPT P10636 4/20 0.52
CYP3A4 P08684 2/20 0.52
MAPK1 P28482 2/20 0.52
TSHR P16473 1/20 0.52
ABCC1 P33527 1/20 0.50
F11 P03951 1/20 0.50
KDM4E B2RXH2 3/20 0.49
HPGD P15428 3/20 0.49
LMNA P02545 2/20 0.49
TP53 P04637 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6314671 0.93 EGFR (0.61) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL6308080 0.92 F11 (0.57) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL7550360 0.91 EGFR (0.53) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL6308755 0.91 EGFR (0.56) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL6315683 0.89 EGFR (0.69) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL6308934 0.89 EGFR (0.64) EGFRPOLBRXFP1MAPTABCC1
SCHEMBL6308357 0.88 EGFR (0.59) EGFRPOLBRXFP1MAPTABCC1
SCHEMBL6314802 0.86 EGFR (0.83) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL6314890 0.85 EGFR (0.86) EGFRPOLBRXFP1ALDH1A1MAPT
SCHEMBL6314294 0.85 EGFR (0.59) EGFRPOLBRXFP1MAPTABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed