SCHEMBL6314671

SCHEMBL6314671

COc1cc(OC)cc(-c2ccc(-c3nc4cc(Cl)ccc4c(=O)n3CCCN)cc2)c1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.61
POLB P06746 4/20 0.54
RXFP1 Q9HBX9 2/20 0.54
ABCC1 P33527 1/20 0.48
MAPT P10636 4/20 0.47
CYP3A4 P08684 1/20 0.47
TP53 P04637 1/20 0.47
F11 P03951 1/20 0.46
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313852 0.93 EGFR (0.64) EGFRPOLBRXFP1ABCC1MAPT
SCHEMBL6315037 0.92 POLB (0.54) EGFRPOLBRXFP1ABCC1MAPT
SCHEMBL6308934 0.88 EGFR (0.64) EGFRPOLBRXFP1ABCC1MAPT
SCHEMBL6309730 0.87 ALDH1A1 (0.59) POLBRXFP1MAPTF11ALDH1A1
SCHEMBL6315683 0.86 EGFR (0.69) EGFRPOLBRXFP1MAPTCYP3A4
SCHEMBL6308755 0.86 EGFR (0.56) EGFRPOLBRXFP1ABCC1MAPT
SCHEMBL6314802 0.85 EGFR (0.83) EGFRPOLBRXFP1MAPTTP53
SCHEMBL6308357 0.85 EGFR (0.59) EGFRPOLBRXFP1ABCC1MAPT
SCHEMBL6314809 0.85 F11 (0.63) POLBRXFP1MAPTF11ALDH1A1
SCHEMBL6308080 0.85 F11 (0.57) EGFRPOLBRXFP1ABCC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed