SCHEMBL6317062

SCHEMBL6317062

Cc1cccc(C[C]=O)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
TAAR1 Q96RJ0 1/20 0.39
TRPA1 O75762 1/20 0.38
ATM Q13315 1/20 0.38
GABRA1 P14867 3/20 0.36
GABRB2 P47870 3/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
CYP3A4 P08684 1/20 0.34
KEAP1 Q14145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1610906 0.83 ESR1 (0.41) ESR1ESR2TAAR1TRPA1ATM
SCHEMBL811980 0.82 TAAR1 (0.52) TAAR1TSHRSMN1; SMN2MAPTGAA
SCHEMBL17077902 0.80 TDP2 (0.32)
SCHEMBL16958334 0.79 ALDH1A1 (0.42) TAAR1GABRA1GABRB2SMN1; SMN2MAPT
SCHEMBL16952334 0.79 GABRA1 (0.38) TAAR1GABRA1GABRB2P2RX7ALDH1A1
SCHEMBL3792645 0.78 ESR1 (0.41) ESR1ESR2TAAR1TRPA1ATM
SCHEMBL8010290 0.77 GABRA1 (0.44) ESR1ESR2TRPA1ATMGABRA1
SCHEMBL29420847 0.77 GABRA1 (0.50) ESR1ESR2TAAR1TRPA1ATM
SCHEMBL140570 0.77 GABRA1 (0.50) ESR1ESR2TAAR1TRPA1ATM
SCHEMBL4094425 0.76 SCN8A (0.37) TAAR1TSHRSMN1; SMN2MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469887-B1 Acetamide derivatives ZENECA LTD (GB) 1994-12-14 EP claimed
US-5270342-A Acetamide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US claimed
EP-0469887-A1 Acetamide derivatives ZENECA LIMITED (GB) 1992-02-05 EP claimed
US-20050158264-A1 Sympathetic nerve-stimulating fragrant compositions SHISEIDO COMPANY, LTD. 2005-07-21 US disclosed
US-20050003976-A1 Sympathetic nerve-stimulating fragrant compositions SHISEIDO COMPANY, LTD. 2005-01-06 US disclosed
EP-1346726-A1 SYMPATHETIC-ACTIVATING PERFUME COMPOSITION SHISEIDO COMPANY, LTD. (JP) 2003-09-24 EP disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
US-5430060-A Aldose reductase inhibitor ZENECA LIMITED (GB) 1995-07-04 US disclosed
EP-0469887-B1 Acetamide derivatives ZENECA LTD (GB) 1994-12-14 EP disclosed
US-5270342-A Acetamide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0469887-A1 Acetamide derivatives ZENECA LIMITED (GB) 1992-02-05 EP disclosed
US-3933806-A Cephalosporin michael adducts ELI LILLY AND COMPANY (US) 1976-01-20 US disclosed