SCHEMBL6317655

SCHEMBL6317655

Cc1c(Cc2ccc(F)cc2F)c(Cl)c2c(nc3ccccn32)c1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.38
HTR2C P28335 3/20 0.38
SMN1; SMN2 Q16637 5/20 0.35
KDM4E B2RXH2 4/20 0.35
RAB9A P51151 3/20 0.35
ADORA1 P30542 1/20 0.34
PIK3CD O00329 3/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PIK3CA P42336 1/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
ENPP2 Q13822 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6312701 0.86 ENPP2 (0.43) SMN1; SMN2KDM4ERAB9AADORA1PIK3CD
SCHEMBL6311410 0.86 PIK3CD (0.38) SMN1; SMN2KDM4EADORA1PIK3CDMEN1
SCHEMBL6311004 0.82 ENPP2 (0.43) SMN1; SMN2KDM4ERAB9AADORA1ENPP2
SCHEMBL6310328 0.81 NPSR1 (0.44) SMN1; SMN2KDM4ERAB9AMEN1KMT2A
SCHEMBL6309849 0.78 KDM4E (0.41) KDM4ERAB9AMEN1KMT2ANPC1
SCHEMBL6312086 0.78 MAPT (0.47) SMN1; SMN2KDM4ERAB9AMEN1KMT2A
SCHEMBL6317979 0.77 ADORA3 (0.43) SMN1; SMN2KDM4ERAB9AADORA1MEN1
SCHEMBL6312786 0.77 KDM4E (0.44) SMN1; SMN2KDM4ERAB9AMEN1KMT2A
SCHEMBL6312626 0.77 PIK3CD (0.45) KDM4ERAB9AADORA1PIK3CDKMT2A
SCHEMBL6311562 0.76 HPGD (0.43) SMN1; SMN2KDM4ERAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050113397-A1 Imidazo[1,2-a]pyridine derivative DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2005-05-26 US disclosed
EP-1479681-A1 IMIDAZO(1,2-a)PYRIDINE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2004-11-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050113397-A1 Imidazo[1,2-a]pyridine derivative MANBA, MAN2B1, ERG28 HTR2A 4490/4885HTR2C 4444/4885SMN1; SMN2 2642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.