SCHEMBL6320255

SCHEMBL6320255

CNC[C@@H](O)c1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.55
CYP3A4 P08684 4/20 0.55
CYP2D6 P10635 4/20 0.55
SLC6A2 P23975 3/20 0.55
SLC6A4 P31645 3/20 0.55
KCNH2 Q12809 2/20 0.55
ADRB3 P13945 6/20 0.53
ADRB1 P08588 5/20 0.53
HIF1A Q16665 4/20 0.53
ADRB2 P07550 4/20 0.53
HTR1A P08908 2/20 0.53
ADRA2A P08913 2/20 0.53
TSHR P16473 2/20 0.53
ADRA2B P18089 2/20 0.53
ADRA2C P18825 2/20 0.53
DRD1 P21728 2/20 0.53
ADRA1A P35348 2/20 0.53
ADRA1B P35368 2/20 0.53
DRD3 P35462 2/20 0.53
NFKB1 P19838 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048311 1.00 SLC6A3 (0.55) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL14126604 0.98 HIF1A (0.54) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
Bromide SCHEMBL6286509 0.98 SLC6A3 (0.53) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL23367359 0.84 SMN1; SMN2 (0.52) SLC6A3SLC6A2SLC6A4ADRB3ADRB1
SCHEMBL10886485 0.83 ADRB1 (0.56) CYP3A4CYP2D6ADRB3ADRB1HIF1A
SCHEMBL30488152 0.83 ADRB1 (0.56) CYP3A4CYP2D6ADRB3ADRB1HIF1A
SCHEMBL25272115 0.83 ADRB1 (0.56) CYP3A4CYP2D6ADRB3ADRB1HIF1A
SCHEMBL23384857 0.81 ADRB3 (0.46) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL16198513 0.81 HTR2A (0.50) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL16198555 0.81 HTR2A (0.50) SLC6A3CYP3A4CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6861438-B2 Antiviral agents PFIZER (US) 2005-03-01 US claimed
EP-1458719-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2004-09-22 EP claimed
US-20040138449-A1 Antiviral agents PHARMACIA & UPJOHN COMPANY 2004-07-15 US claimed
US-20030207877-A1 Pyridoquinoxaline antivirals PHARMACIA & UPJOHN COMPANY 2003-11-06 US claimed
WO-2003053971-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2003-07-03 WO claimed
US-6861438-B2 Antiviral agents PFIZER (US) 2005-03-01 US disclosed
US-6852731-B2 Antiviral compounds PFIZER (US) 2005-02-08 US disclosed
US-20040242884-A1 ANTIVIRAL COMPOUNDS PHARMACIA & UPJOHN COMPANY 2004-12-02 US disclosed
EP-1458719-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2004-09-22 EP disclosed
US-20040138449-A1 Antiviral agents PHARMACIA & UPJOHN COMPANY 2004-07-15 US disclosed
US-20030207877-A1 Pyridoquinoxaline antivirals PHARMACIA & UPJOHN COMPANY 2003-11-06 US disclosed
WO-2003053971-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2003-07-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030207877-A1 Pyridoquinoxaline antivirals IFNAR1, SARS1, ZC3HAV1 SLC6A3 464/4885CYP3A4 601/4885CYP2D6 194/4885
US-20040242884-A1 ANTIVIRAL COMPOUNDS ZC3HAV1, IRF3, IFNAR1 SLC6A3 742/4885CYP3A4 703/4885CYP2D6 1361/4885
US-20040138449-A1 Antiviral agents IRF3, IFNAR1, EIF2AK2 SLC6A3 1295/4885CYP3A4 1526/4885CYP2D6 1364/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.