SCHEMBL6322635

SCHEMBL6322635

CC(C)(C)OC(=O)NCC1CCCN(C(=O)c2ccc3c(Cl)ncnc3c2)C1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
ACACB O00763 4/20 0.44
ACACA Q13085 4/20 0.44
NPC1L1 Q9UHC9 2/20 0.43
EEF2K O00418 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
IRAK1 P51617 1/20 0.42
CNR2 P34972 1/20 0.41
CCRL2 O00421 1/20 0.40
ACKR3 P25106 1/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6331356 0.85 MAP4K4 (0.49) NPC1L1
SCHEMBL6326733 0.82 HCRTR1 (0.41) KMT2AACACBACACANPC1RAB9A
SCHEMBL6330326 0.81 ADORA2A (0.45)
SCHEMBL4150819 0.74 HPGD (0.56) ALDH1A1
SCHEMBL6323082 0.74 HPGD (0.52) KMT2AALDH1A1
SCHEMBL6324733 0.73 HPGD (0.58) ALDH1A1
SCHEMBL4141349 0.72 ACACB (0.40) ACACBACACACCRL2ALDH1A1
SCHEMBL4144760 0.72 ACACB (0.40) ACACBACACACCRL2ALDH1A1
SCHEMBL26230079 0.72 IRAK1 (0.51) ACACBACACAIRAK1CCRL2
SCHEMBL3285436 0.71 PKM (0.61) ACACBACACANPC1L1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050107409-A1 Aromatic bicyclic compounds, preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-05-19 US disclosed
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050107409-A1 Aromatic bicyclic compounds, preparation thereof and their use as pharmaceutical compositions F12, F2, F11 KMT2A 3506/4885ACACB 2102/4885ACACA 639/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.