SCHEMBL6326416

SCHEMBL6326416

CC(C)(CNC(=O)CCCc1nc(-c2ccccc2)no1)CNc1n[nH]c(=O)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
LMNA P02545 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
MAPK1 P28482 1/20 0.50
HTT P42858 1/20 0.50
HDAC1 Q13547 3/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC8 Q9BY41 2/20 0.48
GAA P10253 3/20 0.46
TP53 P04637 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 4/20 0.46
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
TSHR P16473 2/20 0.44
CYP3A4 P08684 1/20 0.44
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6326400 0.95 ALDH1A1 (0.52) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6328351 0.94 GAA (0.51) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6328273 0.94 LMNA (0.48) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6334365 0.94 HDAC1 (0.48) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6331317 0.94 HDAC2 (0.48) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL5073454 0.92 HDAC1 (0.51) ALDH1A1LMNASMN1; SMN2HTTHDAC1
SCHEMBL6328582 0.92 HDAC1 (0.51) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6327916 0.91 NPSR1 (0.43) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6328083 0.90 MAPT (0.48) ALDH1A1LMNASMN1; SMN2MAPK1HTT
SCHEMBL6327919 0.90 HDAC1 (0.42) ALDH1A1LMNASMN1; SMN2MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924284-B2 PARP inhibitors ICOS CORPORATION (US) 2005-08-02 US disclosed