SCHEMBL6329311

SCHEMBL6329311

COc1ccc2c(c1)cc(C)n2S(=O)(=O)c1ccc2c(c1)CNCC2

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PNMT P11086 6/20 0.49
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
HTR6 P50406 4/20 0.44
CYP3A4 P08684 1/20 0.44
KDM4E B2RXH2 2/20 0.42
HTR2C P28335 4/20 0.42
HTR2A P28223 1/20 0.42
TSHR P16473 1/20 0.42
HTR2B P41595 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6330490 0.83 HTR6 (0.61) PNMTADRA2AADRA2BADRA2CHTR6
SCHEMBL6338119 0.79 HTR6 (0.61) PNMTADRA2AADRA2BADRA2CHTR6
SCHEMBL29558442 0.76 HTR2C (0.57) PNMTADRA2AADRA2BADRA2CHTR2C
SCHEMBL746109 0.76 HTR2C (0.57) PNMTADRA2AADRA2BADRA2CHTR2C
Formaldehyde SCHEMBL30554785 0.75 PNMT (0.55) PNMTADRA2AADRA2BADRA2CHTR2C
Hydrochloric Acid SCHEMBL31062521 0.74 HTR2C (0.55) PNMTADRA2AADRA2BADRA2CHTR2C
Hydrochloric Acid SCHEMBL1124555 0.74 HTR2C (0.55) PNMTADRA2AADRA2BADRA2CHTR2C
SCHEMBL3555665 0.74 HTR6 (0.63) HTR6HTR2AMEN1KMT2AL3MBTL1
SCHEMBL6336119 0.72 PNMT (0.60) PNMTADRA2AADRA2BADRA2CHTR6
SCHEMBL6332913 0.71 PNMT (0.53) PNMTADRA2AADRA2BADRA2CHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849644-B2 Isoquinoline derivatives useful in the treatment of CNS disorders SMITHKLINE BEECHAM P.L.C. (GB) 2005-02-01 US claimed