SCHEMBL6330225

SCHEMBL6330225

Cn1ccnc1C#Cc1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.48
GRM5 P41594 6/20 0.45
CHRNB2 P17787 5/20 0.45
CHRNA4 P43681 5/20 0.45
CYP2C9 P11712 3/20 0.45
CYP2B6 P20813 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP2D6 P10635 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2E1 P05181 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C8 P10632 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202593 0.83 HAO1 (0.48) GRM5
SCHEMBL15871038 0.78 LPO (0.48) CHRNB2CHRNA4
SCHEMBL3796332 0.76 CYP2A6 (0.67) CYP2A6GRM5CHRNB2CHRNA4CYP2C9
SCHEMBL6209390 0.73 HAO1 (0.46) GRM5
SCHEMBL13907278 0.72 CYP2A6 (0.62) CYP2A6GRM5CHRNB2CHRNA4CYP2C9
SCHEMBL6208432 0.71 HAO1 (0.53)
SCHEMBL401836 0.70 GRM5 (0.64) CYP2A6GRM5CHRNB2CHRNA4CYP2C9
SCHEMBL31673222 0.70 GRM5 (0.64) CYP2A6GRM5CHRNB2CHRNA4CYP2C9
SCHEMBL31673242 0.69 CYP2A6 (0.58) CYP2A6GRM5CHRNB2CHRNA4CYP2C9
SCHEMBL29993685 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050085523-A1 Imidazolyl and pyrazolyl ethyne compounds COSFORD NICHOLAS D (US) 2005-04-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085523-A1 Imidazolyl and pyrazolyl ethyne compounds CBR3, CBR1, CHRM3 CYP2A6 157/4885GRM5 67/4885CHRNB2 199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.