SCHEMBL633486

SCHEMBL633486

COCc1cccc(N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.52
MAOA P21397 2/20 0.52
CYP19A1 P11511 1/20 0.50
CYP3A4 P08684 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CASP1 P29466 1/20 0.46
RECQL P46063 1/20 0.46
IDO1 P14902 4/20 0.46
AGXT P21549 2/20 0.46
TP53 P04637 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
ACHE P22303 1/20 0.42
ABHD6 Q9BV23 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30601044 1.00 MAOB (0.52) MAOBMAOACYP19A1CYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL6320078 0.98 MAOB (0.53) MAOBMAOACYP19A1CYP3A4ALDH1A1
SCHEMBL487468 0.84 IDO1 (0.48) MAOBCYP3A4IDO1AGXT
SCHEMBL8256843 0.83 MAOB (0.44) MAOBMAOACYP19A1CYP3A4ALDH1A1
SCHEMBL30041293 0.83 MAOB (0.44) MAOBMAOACYP19A1CYP3A4ALDH1A1
SCHEMBL366865 0.82 MAOB (0.56) MAOBMAOACYP19A1CYP3A4ALDH1A1
SCHEMBL1520696 0.80 IDO1 (0.61) MAOBMAOACYP3A4IDO1AGXT
SCHEMBL29684100 0.79 MAOB (0.59) MAOBMAOACYP19A1CYP3A4ALDH1A1
SCHEMBL6678878 0.79 MAOB (0.59) MAOBMAOACYP19A1CYP3A4ALDH1A1
SCHEMBL8011823 0.79 CYP3A4 (0.50) MAOBMAOACYP19A1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 178 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed
US-7678815-B2 Thiazole-4-carboxyamide derivatives HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1844044-A1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2007-10-17 EP claimed
US-20060160857-A1 Thiazole-4-carboxyamide derivatives HOFFMANN-LA ROCHE INC. 2006-07-20 US claimed
WO-2006074884-A1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-07-20 WO claimed
US-4139346-A Nucleic acid and protein binding paper ENZO BIO CHEM INCORPORATED (US) 1979-02-13 US claimed
US-12486258-B2 Compounds and methods for regulating insulin secretion THE BROAD INSTITUTE, INC. (US) 2025-12-02 US disclosed
US-20250115581-A1 SUBSTITUTED PIPERIDINES AS CK1A DEGRADERS MONTE ROSA THERAPEUTICS AG (CH) 2025-04-10 US disclosed
CN-118909239-A Preparation method and application of polyether polyol for adhesive 江苏钟山新材料有限公司 2024-11-08 CN disclosed
CN-114315796-B Compounds used as HPK1 kinase inhibitor, preparation method and application thereof 中国药科大学 2024-03-26 CN disclosed
WO-2023244817-A1 SUBSTITUTED PIPERIDINES AS CK1A DEGRADERS MONTE ROSA THERAPEUTICS, INC. (US) 2023-12-21 WO disclosed
US-20230192607-A1 TRANSCRIPTIONAL ENHANCED ASSOCIATE DOMAIN (TEAD) TRANSCRIPTION FACTOR INHIBITORS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-06-22 US disclosed
US-20230142508-A1 COMPOUNDS AND METHODS FOR REGULATING INSULIN SECRETION THE BROAD INSTITUTE, INC. (US) 2023-05-11 US disclosed
US-4286964-A Polyfunctional epoxides and halohydrins used as bridging groups to bind aromatic amine group-containing alcohols and thiols to hydroxyl bearing substrates SEED BRIAN S 1981-09-01 US disclosed
EP-0027377-A1 Derivatives of hydroxyl-bearing substrates, process for their preparation and a method of application Seed, Brian Sarsfield (US) 1981-04-22 EP disclosed
US-4188371-A CONTACTING RADIOLABELLED ANTISERUM SPECIFIC TO 1,2-PROPANEDIOL DEHYDROGENASE WITH SAMPLE LYSATE, INCUBATING, CONTACTING WITH SOLID PHASE ANTIGEN OR ANTIGEN IMMUNOADSORBENT, INCUBATING, MONITORING CORNING GLASS WORKS (US) 1980-02-12 US disclosed
US-4139346-A Nucleic acid and protein binding paper ENZO BIO CHEM INCORPORATED (US) 1979-02-13 US disclosed
US-4138292-A ENZYMES OR MICROORGANISMS IN A SULFATED POLYSACCHARIDE GEL TANABE SEIYAKU CO., LTD. (JP) 1979-02-06 US disclosed
US-4016043-A Enzymatic immunological method for the determination of antigens and antibodies AKZONA INCORPORATED (US) 1977-04-05 US disclosed
US-RE29169-E PROTEINS, ENZYMES AKZONA INCORPORATED (US) 1977-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230142508-A1 COMPOUNDS AND METHODS FOR REGULATING INSULIN SECRETION IAPP, GPR119, PNLIP MAOB 3316/4885MAOA 3998/4885CYP19A1 2131/4885
US-20060160857-A1 Thiazole-4-carboxyamide derivatives GRM1, GRM2, GRIA4 MAOB 3622/4885MAOA 3677/4885CYP19A1 3116/4885
US-20250115581-A1 SUBSTITUTED PIPERIDINES AS CK1A DEGRADERS CKS1B, CSNK1A1, CKS2 MAOB 4157/4885MAOA 3159/4885CYP19A1 817/4885
US-12486258-B2 Compounds and methods for regulating insulin secretion IAPP, GPR119, PNLIP MAOB 3316/4885MAOA 3998/4885CYP19A1 2131/4885
US-20230192607-A1 TRANSCRIPTIONAL ENHANCED ASSOCIATE DOMAIN (TEAD) TRANSCRIPTION FACTOR INHIBITORS AND USES THEREOF TEAD1, TEAD4, TEAD2 MAOB 3216/4885MAOA 3448/4885CYP19A1 2049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.