SCHEMBL6338355

SCHEMBL6338355

CC(=O)Nc1ccc2c(c1)C(c1cccn1-c1cccc(Cl)c1)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.44
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
AURKB Q96GD4 1/20 0.38
LRRK2 Q5S007 1/20 0.37
MAPT P10636 2/20 0.37
PGR P06401 2/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PTP4A3 O75365 1/20 0.36
RECQL P46063 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDR P35968 1/20 0.35
NOX4 Q9NPH5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6338345 0.92 NQO2 (0.46) NQO2MEN1KMT2ALRRK2MAPT
SCHEMBL11215523 0.73 NQO2 (0.59) NQO2MEN1KMT2AMAPTCHRNB2
SCHEMBL6347633 0.68 PTPN1 (0.32) KMT2AMAPTPGRTDP1
SCHEMBL6988776 0.66 NQO2 (0.51) NQO2MEN1KMT2AMAPTTP53
SCHEMBL357999 0.64 MEN1 (0.71) MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL10059474 0.63 GAA (0.53) NQO2MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL10079113 0.62 FYN (0.45) MEN1KMT2AMAPTSMN1; SMN2NOX4
SCHEMBL18682061 0.62 CHRNB2 (0.57) MEN1KMT2AMAPTTP53TDP1
SCHEMBL11234944 0.60 SMN1; SMN2 (0.63) MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL6815121 0.59 ALDH1A1 (0.70) MEN1KMT2AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6930124-B2 Compounds derived from oxindoles and their therapeutic application in cancer treatment AVENTIS PHARMA S. A. (FR) 2005-08-16 US claimed
US-20040082645-A1 Compounds derived from oxindoles and their therapeutic application in cancer treatment AVENTIS PHARMA S.A. (FR) 2004-04-29 US claimed
US-6930124-B2 Compounds derived from oxindoles and their therapeutic application in cancer treatment AVENTIS PHARMA S. A. (FR) 2005-08-16 US disclosed
US-20040082645-A1 Compounds derived from oxindoles and their therapeutic application in cancer treatment AVENTIS PHARMA S.A. (FR) 2004-04-29 US disclosed
EP-1370555-A1 COMPOUNDS DERIVED FROM OXINDOLES AND THE USE THEREOF IN CANCEROLOGY Aventis Pharma S.A. (FR) 2003-12-17 EP disclosed
WO-2002072575-A1 COMPOUNDS DERIVED FROM OXINDOLES AND THE USE THEREOF IN CANCEROLOGY AVENTIS PHARMA S.A. (FR) 2002-09-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082645-A1 Compounds derived from oxindoles and their therapeutic application in cancer treatment TUBB1, TUBB3, TUBA1C NQO2 806/4885MEN1 1742/4885KMT2A 3941/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.