SCHEMBL6345240

SCHEMBL6345240

COc1ccc2c(c1)C[C@H](C(CCN)CC1CCN(S(C)(=O)=O)CC1)CC2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
ACHE P22303 3/20 0.43
DRD2 P14416 5/20 0.42
DRD3 P35462 5/20 0.42
SIGMAR1 Q99720 3/20 0.41
HTR1A P08908 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
CYP2D6 P10635 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CYP19A1 P11511 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TSHR P16473 1/20 0.38
DRD4 P21917 2/20 0.38
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6335390 1.00 CA1 (0.43) CA1CA2ACHEDRD2DRD3
SCHEMBL6344101 0.96 CA1 (0.43) CA1CA2ACHEDRD2DRD3
SCHEMBL6336495 0.91 ALDH1A1 (0.40) CA1CA2CYP2D6HRH3MEN1
SCHEMBL6334436 0.89 SIGMAR1 (0.44) CA1CA2ACHEDRD2DRD3
SCHEMBL6334414 0.88 CA7 (0.38) CA1CA2MEN1KMT2ATSHR
SCHEMBL6337078 0.87 DPP4 (0.37) CYP2D6HRH3
SCHEMBL6665870 0.87 ALDH1A1 (0.40) CA1CA2CYP2D6HRH3KMT2A
SCHEMBL6342896 0.87 HTR6 (0.42) CA1CA2ACHEDRD2DRD3
SCHEMBL6346802 0.85 CA1 (0.40) CA1CA2ACHEDRD2DRD3
SCHEMBL6338274 0.85 SIGMAR1 (0.44) CA1CA2ACHESIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6864266-B2 4-piperidinyl alkyl amine derivatives as muscarinic receptor antagonists SYNTEX (U.S.A.) LLC (US) 2005-03-08 US claimed