SCHEMBL634722

SCHEMBL634722

NC(=O)c1cccc2c(-c3cccc4c(C(N)=O)cccc34)cccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.55
KMT2A Q03164 1/20 0.55
BCAT2 O15382 1/20 0.54
KDM4E B2RXH2 6/20 0.53
ALDH1A1 P00352 4/20 0.53
GAA P10253 1/20 0.53
KEAP1 Q14145 1/20 0.52
NFE2L2 Q16236 1/20 0.52
HSD17B10 Q99714 2/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
PARP1 P09874 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
METAP2 P50579 1/20 0.45
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GLA P06280 1/20 0.44
NUDT1 P36639 1/20 0.44
PDPK1 O15530 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6135290 0.93 ATM (0.61) ATMKMT2ABCAT2KDM4EALDH1A1
SCHEMBL30646218 0.88 BCAT2 (0.63) ATMKMT2ABCAT2KDM4EALDH1A1
SCHEMBL7916759 0.84 NR4A1 (0.59) ATMKMT2ABCAT2KDM4EALDH1A1
SCHEMBL28639283 0.82 ATM (0.75) ATMKMT2ABCAT2KDM4EALDH1A1
SCHEMBL6061358 0.82 ALDH1A1 (0.56) ATMKMT2AKDM4EALDH1A1GAA
SCHEMBL4134419 0.82 KDM4E (0.61) ATMKMT2AKDM4EALDH1A1GAA
SCHEMBL30892682 0.81 BCAT2 (0.55) KMT2ABCAT2KDM4EALDH1A1GAA
SCHEMBL5849850 0.81 BCAT2 (0.55) KMT2ABCAT2KDM4EALDH1A1GAA
SCHEMBL31621277 0.81 BCAT2 (0.55) KMT2ABCAT2KDM4EALDH1A1GAA
SCHEMBL5772703 0.80 PRNP (0.58) ATMKMT2AKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418942-A1 NAPHTHALENE-BASED INHIBITORS OF ANTI-APOPTOTIC PROTEINS Sanford-Burnham Medical Research Institute (US) 2012-02-22 EP disclosed
WO-2010120943-A1 NAPHTHALENE-BASED INHIBITORS OF ANTI-APOPTOTIC PROTEINS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2010-10-21 WO disclosed