SCHEMBL9602391

SCHEMBL9602391

CN1C2CCC1CC(NC(=O)ON1CC(C)(C)c3ccccc31)C2

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NOTUM Q6P988 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ricasetron SCHEMBL21715163 0.81 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL634827 0.81 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL634826 0.81 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL20362251 0.81 NOTUM (0.52) NOTUM
Ricasetron SCHEMBL7445859 0.81 NOTUM (0.51) NOTUM
SCHEMBL9602248 0.77 MEN1 (0.43) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL9602684 0.76 HTR6 (0.46) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL9602968 0.76 CHRM2 (0.50)
SCHEMBL7346340 0.74 TMEM97 (0.48)
SCHEMBL9601595 0.73 TMEM97 (0.43) MEN1KMT2AALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0247266-B1 INDOLE DERIVATIVES HAVING AN AZABICYCLIC SIDE CHAIN, PROCESS FOR THEIR PREPARATION, INTERMEDIATES, AND PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1993-03-10 EP claimed