SCHEMBL6349253

SCHEMBL6349253

CCCCOC(C)Oc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCCOC4)cc2)CCN3C(=O)CC2(C)OCCO2)cc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.42
CCR5 P51681 15/20 0.36
CCR7 P32248 1/20 0.36
HDAC1 Q13547 1/20 0.35
CCR3 P51677 1/20 0.35
CCR4 P51679 1/20 0.35
CXCR5 P32302 1/20 0.33
CXCR3 P49682 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486829 0.91 CCR5 (0.44) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6338777 0.87 CCR2 (0.47) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6341948 0.87 CCR2 (0.51) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6342701 0.87 MAPT (0.43) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6339722 0.84 CCR2 (0.48) CCR2CCR5CCR7CCR3CCR4
SCHEMBL6342647 0.84 CCR2 (0.51) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6350471 0.83 CCR2 (0.45) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6350329 0.83 CCR2 (0.49) CCR2CCR5CCR7HDAC1CXCR5
SCHEMBL6340354 0.82 CCR2 (0.44) CCR2CCR5CCR7HDAC1CCR3
SCHEMBL6341367 0.82 CCR5 (0.44) CCR2CCR5CCR7HDAC1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed