SCHEMBL6350329

SCHEMBL6350329

CCCCOC(C)Oc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCCOC4)cc2)CCN3)cc1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.49
HDAC1 Q13547 1/20 0.40
CCR5 P51681 15/20 0.39
CXCR3 P49682 3/20 0.39
CCR7 P32248 2/20 0.39
CXCR5 P32302 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6350327 0.90 CCR2 (0.51) CCR2HDAC1CCR5CXCR3CCR7
SCHEMBL6338777 0.86 CCR2 (0.47) CCR2HDAC1CCR5CCR7
SCHEMBL6341948 0.86 CCR2 (0.51) CCR2HDAC1CCR5CCR7
SCHEMBL6339722 0.83 CCR2 (0.48) CCR2CCR5CCR7
SCHEMBL6342647 0.83 CCR2 (0.51) CCR2HDAC1CCR5CCR7
SCHEMBL6342701 0.83 MAPT (0.43) CCR2HDAC1CCR5CCR7
SCHEMBL6349253 0.83 CCR2 (0.42) CCR2HDAC1CCR5CXCR3CCR7
SCHEMBL6350471 0.82 CCR2 (0.45) CCR2HDAC1CCR5CXCR3CCR7
SCHEMBL6341780 0.82 CCR2 (0.58) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL6340354 0.81 CCR2 (0.44) CCR2HDAC1CCR5CXCR3CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed