SCHEMBL6349338

SCHEMBL6349338

CCCN1CCC(C(=O)Nc2ccc(CN(C)C3CCOCC3)cc2)=Cc2cc(-c3ccc(N4CCOCC4)cc3)ccc21

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.60
CCR5 P51681 15/20 0.50
MCHR1 Q99705 1/20 0.43
CXCR3 P49682 3/20 0.42
CCR7 P32248 2/20 0.42
CXCR5 P32302 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6340391 0.89 CCR2 (0.61) CCR2CCR5MCHR1CXCR3CCR7
SCHEMBL6353376 0.88 CCR2 (0.60) CCR2CCR5MCHR1CXCR3CCR7
SCHEMBL6340461 0.88 CCR2 (0.59) CCR2CCR5MCHR1CXCR3CCR7
SCHEMBL6351839 0.88 CCR2 (0.59) CCR2CCR5MCHR1CXCR3CCR7
SCHEMBL5205469 0.87 CCR2 (0.63) CCR2CCR5MCHR1CXCR3CCR7
SCHEMBL6341093 0.87 CCR2 (0.54) CCR2CCR5CXCR3CCR7
SCHEMBL6344086 0.87 CCR2 (0.57) CCR2CCR5CCR7
SCHEMBL6350296 0.87 CCR2 (0.55) CCR2CCR5CCR7
SCHEMBL6340941 0.87 CCR5 (0.58) CCR2CCR5CCR7
Hydrochloric Acid SCHEMBL6350443 0.86 CCR5 (0.57) CCR2CCR5CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed