Estramustine

Estramustine

SCHEMBL6353316

C[C@]12CC[C@@H]3c4ccc(OC(=O)N(CCCl)CCCl)cc4CC[C@H]3[C@@H]1CCC2O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 2/20 1.00
BLM P54132 2/20 1.00
ESR1 P03372 6/20 0.76
ADORA3 P0DMS8 3/20 0.76
INPPL1 O15357 1/20 0.76
PTPN1 P18031 1/20 0.76
DRD1 P21728 1/20 0.76
PTPN6 P29350 1/20 0.76
KDR P35968 1/20 0.76
PTPN11 Q06124 1/20 0.76
LMNA P02545 5/20 0.73
SMN1; SMN2 Q16637 3/20 0.73
ATM Q13315 2/20 0.73
PGR P06401 2/20 0.73
AR P10275 2/20 0.73
SLC6A3 Q01959 2/20 0.73
CHRM1 P11229 1/20 0.73
TBXA2R P21731 1/20 0.73
ADRA1A P35348 1/20 0.73
OPRM1 P35372 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Estramustine SCHEMBL2348477 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL8173336 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL14031683 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL4252 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL29349776 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL29374661 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL13753350 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL7200287 1.00 RECQL (1.00) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL679202 0.99 RECQL (0.98) RECQLBLMESR1ADORA3INPPL1
Estramustine SCHEMBL7621246 0.99 RECQL (0.98) RECQLBLMESR1ADORA3INPPL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6838469-B2 Pharmaceutical composition that exhibits reduced side-effects comprising O-(3-piperidino-2-hydroxy-1-propyl)nicotinic acid amidoxime and a pyrimidine derivative with known antitumor activity N-GENE RESEARCH LABORATORIES INC. (US) 2005-01-04 US disclosed
WO-2004045611-A1 USE OF A THIAZOLIDINEDIONE FOR THE REDUCTION OF SIDE EFFECTS OF CHEMOTHERAPY N-GENE RESEARCH LABORATORIES INC. (US) 2004-06-03 WO disclosed
EP-0993304-B1 PHARMACEUTICAL COMPOSITION HAVING ENHANCED ANTITUMOR ACTIVITY AND/OR REDUCED SIDE EFFECTS, CONTAINING AN ANTITUMOR AGENT AND AN HYDROXAMIC ACID DERIVATIVE N GENE RES LAB INC (US) 2003-04-02 EP disclosed
US-20030050345-A1 Pharmaceutical composition having enhanced antitumor activity and/or reduced side effects, containing an antitumor agent and an hydroximic acid derivative N-GENE RESEARCH LABORATORIES, INC. 2003-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030050345-A1 Pharmaceutical composition having enhanced antitumor activity and/or reduced side effects, containing an antitumor agent and an hydroximic acid derivative H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HDGF, CA7 RECQL 3073/4885BLM 4035/4885ESR1 4870/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.