SCHEMBL6359035

SCHEMBL6359035

Cn1cc(C(=O)Nc2ccc3cccnc3c2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.57
MAOB P27338 3/20 0.54
CNR2 P34972 2/20 0.53
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
CNR1 P21554 1/20 0.52
S1PR1 P21453 4/20 0.52
S1PR3 Q99500 4/20 0.52
TRPV1 Q8NER1 1/20 0.49
CMA1 P23946 1/20 0.47
P2RY14 Q15391 1/20 0.47
NOTUM Q6P988 1/20 0.47
CYP2C9 P11712 1/20 0.47
AURKA O14965 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6359316 0.82 CNR2 (0.53) CNR2KMT2AMEN1CNR1TRPV1
SCHEMBL3879676 0.78 GRM4 (0.64) KMT2AMEN1NPC1RAB9ATRPV1
SCHEMBL3891697 0.77 MEN1 (0.62) KMT2AMEN1NPC1RAB9ATRPV1
SCHEMBL6005094 0.76 MAOB (0.61) HTR2CMAOBKMT2ANPC1
SCHEMBL9165502 0.76 HTR2C (0.61) HTR2CMAOBKMT2AMEN1NPC1
SCHEMBL2661003 0.76 NPC1 (0.83) HTR2CKMT2AMEN1NPC1RAB9A
SCHEMBL18132530 0.76 MEN1 (0.61) KMT2AMEN1NPC1RAB9ATRPV1
SCHEMBL7101847 0.74 PABPC1 (0.79) KMT2AMEN1NPC1RAB9ATRPV1
SCHEMBL29176621 0.74 MAOB (0.62) MAOBKMT2AMEN1AURKA
SCHEMBL4811502 0.74 MAOB (0.84) MAOBKMT2AMEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050165049-A1 Vanilloid receptor ligands and their use in treatments AMGEN, INC. 2005-07-28 US claimed
US-7544803-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2009-06-09 US disclosed
US-7544803-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2009-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165049-A1 Vanilloid receptor ligands and their use in treatments TRPV1, TRPV2, TRPV3 HTR2C 156/4885MAOB 1213/4885CNR2 171/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.