SCHEMBL6368183

SCHEMBL6368183

CCOC(=O)NN[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
MMP8 P22894 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
CTSL P07711 2/20 0.47
TACR1 P25103 1/20 0.47
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
MME P08473 3/20 0.46
POLB P06746 2/20 0.46
ACE P12821 1/20 0.46
CPA1 P15085 1/20 0.46
ACE2 Q9BYF1 1/20 0.46
RAB9A P51151 1/20 0.45
ALDH1A1 P00352 1/20 0.45
ALOX15 P16050 1/20 0.45
ATM Q13315 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368188 1.00 GAA (0.53) GAAMMP8L3MBTL1CTSLTACR1
SCHEMBL6703453 0.88 TACR1 (0.56) CTSLTACR1CTSBCTSSCTSK
SCHEMBL6703452 0.88 TACR1 (0.56) CTSLTACR1CTSBCTSSCTSK
SCHEMBL6367145 0.86 MMP2 (0.46) CTSLCTSBCTSSCTSKMME
SCHEMBL6367149 0.86 MMP2 (0.46) CTSLCTSBCTSSCTSKMME
SCHEMBL3769914 0.85 L3MBTL1 (0.58) MMP8L3MBTL1CTSLCTSBCTSS
SCHEMBL996291 0.85 L3MBTL1 (0.58) MMP8L3MBTL1CTSLCTSBCTSS
SCHEMBL996293 0.85 L3MBTL1 (0.58) MMP8L3MBTL1CTSLCTSBCTSS
Hydrochloric Acid SCHEMBL28046933 0.84 L3MBTL1 (0.57) MMP8L3MBTL1CTSLCTSBCTSS
Hydrochloric Acid SCHEMBL27371193 0.84 L3MBTL1 (0.57) MMP8L3MBTL1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US disclosed