Ebalzotan

Ebalzotan

SCHEMBL6370473

CCCN(C(C)C)C1COc2cccc(C(=O)NC(C)C)c2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ebalzotan SCHEMBL247755 1.00 DRD2 (0.77) DRD2
Hydrochloric Acid SCHEMBL8823814 0.90 DRD2 (0.77) DRD2
Hydrochloric Acid SCHEMBL8823793 0.89 DRD2 (0.76) DRD2
SCHEMBL9568770 0.89 DRD2 (0.76) DRD2
SCHEMBL8823678 0.88 DRD2 (0.78) DRD2
SCHEMBL8823628 0.88 DRD2 (0.78) DRD2
SCHEMBL8823789 0.87 DRD2 (0.76) DRD2
SCHEMBL8823704 0.87 DRD2 (0.58) DRD2
SCHEMBL8823697 0.87 DRD2 (0.58) DRD2
SCHEMBL8823639 0.86 DRD2 (0.82) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5656658-A Method for the treatment of anxiety ASTRA AKTIEBOLAG (SE) 1997-08-12 US claimed
US-5641807-A Method for the treatment of depression ASTRA AKTIEBOLAG (SE) 1997-06-24 US claimed
US-5639784-A ADMINISTERING 3-AMINO-5-CARBAMOYL-CHROMENES AND DERIVATIVES ASTRA AKTIEBOLAG (SE) 1997-06-17 US claimed
EP-0607274-B1 3-(N-ISOPROPYL-N-n-PROPYLAMINO)-5-(N-ISOPROPYL)CARBAMOYLCHROMAN ASTRA AB (SE) 1996-06-26 EP claimed
US-5420151-A Chroman derivatives AKTIEBOLAGET ASTRA (SE) 1995-05-30 US claimed
EP-0538222-A1 3-(N-Isopropyl-N-n-propylamino)-5-(N-isopropyl)carbamoylchroman as a selective 5-hydroxytryptamine receptor stimulant Astra Aktiebolag (SE) 1993-04-21 EP claimed
US-20050004105-A1 Treatment for a attention-deficit hyperactivity disorder PSYCHOGENCIS, INC. 2005-01-06 US disclosed
WO-2004069339-A1 TREATMENT FOR ATTENTION-DEFICIT HYPERACTIVITY DISORDER PSYCHOGENICS INC. (US) 2004-08-19 WO disclosed
US-5656657-A Chroman derivatives ASTRA AKTIEBOLAG (SE) 1997-08-12 US disclosed
US-5656658-A Method for the treatment of anxiety ASTRA AKTIEBOLAG (SE) 1997-08-12 US disclosed
US-5650524-A Process for preparing (R)-3-amino-5-methoxychroman ASTRA AKTIEBOLAG (SE) 1997-07-22 US disclosed
US-5646309-A Intermediates in the synthesis of chroman derivatives ASTRA AKTIEBOLAG (SE) 1997-07-08 US disclosed
US-5641807-A Method for the treatment of depression ASTRA AKTIEBOLAG (SE) 1997-06-24 US disclosed
EP-0607274-A1 3-(N-ISOPROPYL-N-n-PROPYLAMINO)-5-(N-ISOPROPYL)CARBAMOYLCHROMAN. ASTRA AB (SE) 1994-07-27 EP disclosed
EP-0538222-A1 3-(N-Isopropyl-N-n-propylamino)-5-(N-isopropyl)carbamoylchroman as a selective 5-hydroxytryptamine receptor stimulant Astra Aktiebolag (SE) 1993-04-21 EP disclosed
EP-0538222-A1 3-(N-Isopropyl-N-n-propylamino)-5-(N-isopropyl)carbamoylchroman as a selective 5-hydroxytryptamine receptor stimulant Astra Aktiebolag (SE) 1993-04-21 EP disclosed
EP-0538222-A1 3-(N-Isopropyl-N-n-propylamino)-5-(N-isopropyl)carbamoylchroman as a selective 5-hydroxytryptamine receptor stimulant Astra Aktiebolag (SE) 1993-04-21 EP disclosed
WO-1993007135-A1 3-(N-ISOPROPYL-N-N-PROPYLAMINO)-5-(N-ISOPROPYL)CARBAMOYLCHROMAN AKTIEBOLAGET ASTRA (SE) 1993-04-15 WO disclosed
WO-1993007135-A1 3-(N-ISOPROPYL-N-N-PROPYLAMINO)-5-(N-ISOPROPYL)CARBAMOYLCHROMAN AKTIEBOLAGET ASTRA (SE) 1993-04-15 WO disclosed
WO-1993007135-A1 3-(N-ISOPROPYL-N-N-PROPYLAMINO)-5-(N-ISOPROPYL)CARBAMOYLCHROMAN AKTIEBOLAGET ASTRA (SE) 1993-04-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004105-A1 Treatment for a attention-deficit hyperactivity disorder HTR1A, HTR5A, HTR2A DRD2 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.