SCHEMBL6371190

SCHEMBL6371190

CC1Cc2cc([N+](=O)[O-])ccc2NC1=O

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.50
ADRA2A P08913 3/20 0.50
ADRA2B P18089 3/20 0.50
ADRA2C P18825 3/20 0.50
ALDH1A1 P00352 5/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
PGR P06401 2/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CHRNA7 P36544 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
TDP2 O95551 1/20 0.44
CAPN9 O14815 1/20 0.44
CASP3 P42574 1/20 0.44
GAA P10253 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30100720 1.00 PNMT (0.50) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL27377888 0.82 PNMT (0.50) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL1347469 0.81 BRD4 (0.55) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL13007537 0.78 SIRT2 (0.45) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL257552 0.77 ALDH1A1 (0.62) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL6968655 0.77 ALDH1A1 (0.62) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL18743294 0.76 ACHE (0.49) ALDH1A1
SCHEMBL434007 0.76 ACHE (0.49) ALDH1A1
SCHEMBL16333559 0.76 ALDH1A1 (0.42) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL14550603 0.75 BRD4 (0.51) PNMTADRA2AADRA2BADRA2CMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230128402-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF THE TRUSTEES OF PRINCETON UNIVERSITY 2023-04-27 US disclosed
US-20230128402-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF THE TRUSTEES OF PRINCETON UNIVERSITY 2023-04-27 US disclosed
WO-2021151062-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF THE TRUSTEES OF PRINCETON UNIVERISTY (US) 2021-07-29 WO disclosed
WO-2013027168-A1 NOVEL HETEROCYCLIC COMPOUNDS AS BROMODOMAIN INHIBITORS PFIZER INC. (US) 2013-02-28 WO disclosed
US-20050165006-A1 Quinoline derivatives, their preparation and pharmaceutical compositions comprising the same HYUNDAI PHARM. IND. CO., LTD. (KR) 2005-07-28 US disclosed
WO-2003082286-A1 QUINOLINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHEMON INC. (KR) 2003-10-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165006-A1 Quinoline derivatives, their preparation and pharmaceutical compositions comprising the same SLC18A2, SLC6A4, SLC6A2 PNMT 323/4885ADRA2A 274/4885ADRA2B 246/4885
US-20230128402-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PAH, ALDH2, IDH2 PNMT 1641/4885ADRA2A 1558/4885ADRA2B 1154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.