SCHEMBL6373371

SCHEMBL6373371

O=C(O)[C@H](Cc1ccc(O)c(I)c1)NC(=O)[C@@H]1SCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.47
ITGB1 P05556 9/20 0.47
ITGB7 P26010 6/20 0.47
FOLH1 Q04609 2/20 0.43
ALB P02768 2/20 0.40
IL2 P60568 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6367618 0.91 ITGA4 (0.46) ITGA4ITGB1ITGB7
SCHEMBL6367240 0.89 ITGA4 (0.51) ITGA4ITGB1ITGB7
SCHEMBL6372390 0.85 ITGA4 (0.51) ITGA4ITGB1ITGB7
SCHEMBL6373309 0.84 ITGA4 (0.63) ITGA4ITGB1ITGB7
SCHEMBL6375296 0.81 ITGA4 (0.54) ITGA4ITGB1ITGB7
SCHEMBL6373870 0.79 ITGA4 (0.53) ITGA4ITGB1ITGB7
SCHEMBL6373490 0.77 ITGB1 (0.66) ITGA4ITGB1ITGB7
SCHEMBL6368571 0.77 ITGA4 (0.51) ITGA4ITGB1ITGB7
SCHEMBL6368438 0.75 ITGA4 (0.69) ITGA4ITGB1ITGB7
SCHEMBL6368962 0.74 ITGB1 (0.61) ITGA4ITGB1ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed