SCHEMBL6367240

SCHEMBL6367240

O=C(O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H]1SCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.51
ITGB1 P05556 9/20 0.51
ITGB7 P26010 6/20 0.51
ITGA5 P08648 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CCKBR P32239 1/20 0.41
HSD11B1 P28845 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6375296 0.92 ITGA4 (0.54) ITGA4ITGB1ITGB7ITGA5HSD11B1
SCHEMBL6373371 0.89 ITGA4 (0.47) ITGA4ITGB1ITGB7
SCHEMBL6372390 0.88 ITGA4 (0.51) ITGA4ITGB1ITGB7CA2CCKBR
SCHEMBL6367618 0.87 ITGA4 (0.46) ITGA4ITGB1ITGB7HSD11B1
SCHEMBL6368457 0.85 ITGA4 (0.48) ITGA4ITGB1ITGB7ITGA5CA1
SCHEMBL6373870 0.84 ITGA4 (0.53) ITGA4ITGB1ITGB7ITGA5HSD11B1
SCHEMBL6368456 0.83 ITGA4 (0.70) ITGA4ITGB1ITGB7ITGA5
SCHEMBL6368571 0.82 ITGA4 (0.51) ITGA4ITGB1ITGB7ITGA5
SCHEMBL3385855 0.80 ALDH1A1 (0.54) ITGA4ITGB1ITGB7ITGA5
SCHEMBL6368647 0.79 HSD11B1 (0.50) ITGA4ITGB1ITGB7ITGA5CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed