SCHEMBL6368571

SCHEMBL6368571

O=C(O)[C@H](Cc1ccc(OS(=O)(=O)O)cc1)NC(=O)[C@@H]1SCCN1S(=O)(=O)c1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 15/20 0.51
ITGB1 P05556 11/20 0.51
ITGB7 P26010 6/20 0.50
ITGA5 P08648 2/20 0.41
PTPN11 Q06124 1/20 0.40
GPR34 Q9UPC5 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6375296 0.90 ITGA4 (0.54) ITGA4ITGB1ITGB7ITGA5PTPN11
SCHEMBL6373870 0.89 ITGA4 (0.53) ITGA4ITGB1ITGB7ITGA5PTPN11
SCHEMBL6367911 0.82 ITGA4 (0.53) ITGA4ITGB1ITGB7
SCHEMBL6367240 0.82 ITGA4 (0.51) ITGA4ITGB1ITGB7ITGA5
SCHEMBL6368647 0.81 HSD11B1 (0.50) ITGA4ITGB1ITGB7ITGA5
SCHEMBL6372390 0.81 ITGA4 (0.51) ITGA4ITGB1ITGB7
SCHEMBL6368956 0.80 HSD11B1 (0.45) ITGA4ITGB1ITGB7ITGA5GPR34
SCHEMBL6374122 0.78 HSD11B1 (0.47) ITGA4ITGB1ITGB7ITGA5
SCHEMBL6367279 0.78 LMNA (0.45) ITGA4ITGB1ITGB7ITGA5
SCHEMBL3385855 0.77 ALDH1A1 (0.54) ITGA4ITGB1ITGB7ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed